SCHEMBL28051137

SCHEMBL28051137

COc1cc(NS(=O)(=O)c2ccc3c(c2)c2ccccc2n3C)cc(OC)c1OC

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTT P42858 4/20 0.61
SMN1; SMN2 Q16637 2/20 0.61
MAPT P10636 3/20 0.50
TP53 P04637 1/20 0.50
THRB P10828 1/20 0.50
ALDH1A1 P00352 4/20 0.48
CA12 O43570 1/20 0.48
CA9 Q16790 1/20 0.48
PDE3A Q14432 1/20 0.47
PKM P14618 3/20 0.47
L3MBTL1 Q9Y468 2/20 0.47
LMNA P02545 3/20 0.47
RXFP1 Q9HBX9 1/20 0.47
MITF O75030 1/20 0.46
KEAP1 Q14145 1/20 0.46
NFE2L2 Q16236 1/20 0.46
KDM4E B2RXH2 2/20 0.46
HPGD P15428 2/20 0.46
HSD17B10 Q99714 2/20 0.46
MEN1 O00255 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23148487 0.88 MAPT (0.61) HTTSMN1; SMN2MAPTTP53THRB
SCHEMBL28298620 0.87 HTT (0.57) HTTSMN1; SMN2MAPTTP53THRB
SCHEMBL28051052 0.82 ALDH1A1 (0.53) HTTSMN1; SMN2MAPTTP53ALDH1A1
SCHEMBL27651555 0.79 ALDH1A1 (0.54) HTTSMN1; SMN2MAPTTP53THRB
SCHEMBL27651556 0.79 ALDH1A1 (0.60) HTTMAPTTP53THRBALDH1A1
SCHEMBL6073370 0.77 CA12 (0.59) HTTSMN1; SMN2MAPTALDH1A1CA12
SCHEMBL31687144 0.76 HTT (0.55) HTTSMN1; SMN2MAPTTP53THRB
SCHEMBL26792 0.76 PKM (0.61) HTTSMN1; SMN2MAPTTP53THRB
SCHEMBL31687177 0.76 IMPDH2 (0.54) HTTSMN1; SMN2MAPTTP53THRB
SCHEMBL28051135 0.76 HTT (0.52) HTTSMN1; SMN2MAPTTP53THRB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105287388-B High dispersive carbazole sulfonamide derivative and preparation method thereof 山西普德药业有限公司 2019-09-17 CN claimed
CN-105418487-B Carbazole sulfonamide derivative eutectic and preparation method thereof 山西普德药业有限公司 2018-11-02 CN claimed
CN-105418487-A Carbazole sulfonamide derivative eutectic and preparation method thereof SHANXI PUDE PHARMACEUTICS CO LTD 2016-03-23 CN claimed
CN-105287388-A High-dispersion carbazole sulfonamide derivatives and preparation method thereof SHANXI PUDE PHARMACEUTICS CO LTD 2016-02-03 CN claimed
CN-105287388-B High dispersive carbazole sulfonamide derivative and preparation method thereof 山西普德药业有限公司 2019-09-17 CN disclosed
CN-105418487-B Carbazole sulfonamide derivative eutectic and preparation method thereof 山西普德药业有限公司 2018-11-02 CN disclosed
CN-105418487-A Carbazole sulfonamide derivative eutectic and preparation method thereof SHANXI PUDE PHARMACEUTICS CO LTD 2016-03-23 CN disclosed
CN-105287388-A High-dispersion carbazole sulfonamide derivatives and preparation method thereof SHANXI PUDE PHARMACEUTICS CO LTD 2016-02-03 CN disclosed