SCHEMBL28052294

SCHEMBL28052294

Cc1cnn(Cc2ccc(CC(Cc3c[nH]nc3C3CC3)OC=O)cc2)c1

nearest known ligand 0.40

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
KLKB1 P03952 18/20 0.40
NPC1 O15118 1/20 0.31
RAB9A P51151 1/20 0.31
SMN1; SMN2 Q16637 1/20 0.31
PTGER4 P35408 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28052170 0.77 KLKB1 (0.35) KLKB1
SCHEMBL28825964 0.71 CHRNB2 (0.32)
SCHEMBL28052255 0.67 KLKB1 (0.36) KLKB1
SCHEMBL17229326 0.65 KLKB1 (0.46) KLKB1
SCHEMBL16247156 0.65 KLKB1 (0.59) KLKB1
SCHEMBL16486803 0.64 KLKB1 (0.48) KLKB1RAB9ASMN1; SMN2
SCHEMBL16246833 0.64 KLKB1 (0.56) KLKB1NPC1
SCHEMBL17685596 0.63 NPC1 (0.74) KLKB1NPC1RAB9ASMN1; SMN2
SCHEMBL15759268 0.63 KLKB1 (0.51) KLKB1NPC1RAB9ASMN1; SMN2
SCHEMBL26946141 0.62 GABRA1 (0.30)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105452240-A Heterocyclic derivates KALVISTA PHARMACEUTICALS LTD 2016-03-30 CN disclosed