SCHEMBL28052874

SCHEMBL28052874

O=C(Cl)c1c(F)ccc(Br)c1F

nearest known ligand 0.38

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.38
ALOX15 P16050 1/20 0.38
CES2 O00748 4/20 0.37
CES1 P23141 4/20 0.37
NPC1 O15118 2/20 0.33
RAB9A P51151 2/20 0.33
KDM1A O60341 2/20 0.32
KCNH2 Q12809 2/20 0.32
KDM1B Q8NB78 2/20 0.32
LMNA P02545 1/20 0.32
HPGD P15428 1/20 0.31
SMN1; SMN2 Q16637 1/20 0.31
PLAU P00749 1/20 0.31
ELANE P08246 1/20 0.31
KIF11 P52732 1/20 0.31
HTT P42858 1/20 0.31
CA1 P00915 1/20 0.30
CA2 P00918 1/20 0.30
CA4 P22748 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1022860 0.82 CES2 (0.46) ALDH1A1ALOX15CES2CES1LMNA
SCHEMBL671154 0.81 CES2 (0.38) CES2CES1LMNASMN1; SMN2PLAU
SCHEMBL29975604 0.81 CES2 (0.38) CES2CES1LMNASMN1; SMN2PLAU
SCHEMBL16936918 0.80 ALDH1A1 (0.33) ALDH1A1ALOX15KDM1AKCNH2KDM1B
SCHEMBL16555805 0.79 DGAT1 (0.41) CES2CES1NPC1RAB9AKDM1A
SCHEMBL30632655 0.79 DGAT1 (0.41) CES2CES1NPC1RAB9AKDM1A
SCHEMBL10325437 0.79 CES2 (0.37) CES2CES1LMNAHPGDPLAU
SCHEMBL1197627 0.78 ALDH1A1 (0.48) ALDH1A1ALOX15CES2CES1HPGD
SCHEMBL18797709 0.78 ALDH1A1 (0.39) ALDH1A1ALOX15CES2CES1NPC1
SCHEMBL15809161 0.75 CES2 (0.52) ALDH1A1ALOX15CES2CES1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109071457-A Inhibitors of indoleamine 2, 3-dioxygenase 荷兰转化研究中心有限责任公司 2018-12-21 CN disclosed
CN-108473481-A compounds useful as kinase inhibitors 洛克索肿瘤学股份有限公司 2018-08-31 CN disclosed
CN-105683164-A Fungicidal pyrazoles 杜邦公司 2016-06-15 CN disclosed