SCHEMBL28053322

SCHEMBL28053322

NS(=O)(=O)c1cncc(-c2cncc(Cl)c2O)c1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
APLNR P35414 1/20 0.51
PIK3CG P48736 2/20 0.39
PIK3CD O00329 1/20 0.39
PTGS1 P23219 2/20 0.37
PTGS2 P35354 2/20 0.37
CA1 P00915 7/20 0.36
CA2 P00918 7/20 0.36
CA9 Q16790 6/20 0.36
VRK2 Q86Y07 1/20 0.36
CDK2 P24941 1/20 0.35
CA12 O43570 3/20 0.35
CA7 P43166 2/20 0.34
CA14 Q9ULX7 2/20 0.34
IKBKB O14920 1/20 0.34
CHUK O15111 1/20 0.34
LMNA P02545 2/20 0.33
POLB P06746 2/20 0.33
ALDH1A1 P00352 1/20 0.33
CYP2C9 P11712 1/20 0.33
CA4 P22748 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28053327 0.89 APLNR (0.45) APLNRPTGS1PTGS2CA1CA2
SCHEMBL28053258 0.78 PKM (0.46) APLNRPTGS1PTGS2CA1CA2
SCHEMBL28053345 0.78 APLNR (0.50) APLNRPIK3CGPIK3CDPTGS1PTGS2
SCHEMBL28053242 0.77 APLNR (0.43) APLNRPTGS1PTGS2CA1CA2
SCHEMBL28053347 0.75 CA1 (0.44) APLNRPTGS1PTGS2CA1CA2
SCHEMBL28053374 0.74 LRRK2 (0.44) APLNRPIK3CGPIK3CDPTGS1PTGS2
SCHEMBL28826183 0.74 APLNR (0.40) APLNRPTGS1PTGS2CA1CA2
SCHEMBL28053239 0.72 APLNR (0.38) APLNRPTGS1PTGS2CA1CA2
SCHEMBL28053310 0.72 SCN10A (0.44) APLNRCA1CA2CA9CA12
SCHEMBL28826194 0.70 SOS1 (0.39) APLNRCA1CA2CA9CA12

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105377837-A N-(heteroaryl)-sulfonamide derivatives useful as S100-inhibitors ACTIVE BIOTECH AB 2016-03-02 CN claimed
CN-105377837-A N-(heteroaryl)-sulfonamide derivatives useful as S100-inhibitors ACTIVE BIOTECH AB 2016-03-02 CN disclosed