SCHEMBL28053799

SCHEMBL28053799

Cc1nc(C)c(C=Cc2ccccc2)nc1C

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GRM4 Q14833 7/20 0.56
P2RX3 P56373 1/20 0.54
ALDH1A1 P00352 7/20 0.50
KDM4E B2RXH2 7/20 0.50
HPGD P15428 4/20 0.50
RAB9A P51151 5/20 0.48
MEN1 O00255 4/20 0.48
KMT2A Q03164 4/20 0.48
NPC1 O15118 4/20 0.48
SMN1; SMN2 Q16637 3/20 0.48
GRM5 P41594 1/20 0.48
NPSR1 Q6W5P4 1/20 0.48
HDAC6 Q9UBN7 1/20 0.48
CYP3A4 P08684 1/20 0.48
CYP2D6 P10635 1/20 0.48
CYP2C9 P11712 1/20 0.48
PKM P14618 1/20 0.48
TSHR P16473 1/20 0.48
NFKB1 P19838 1/20 0.48
CYP2C19 P33261 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28053933 0.88 MAOB (0.54) GRM4P2RX3ALDH1A1KDM4EHPGD
SCHEMBL28053802 0.82 ALOX5 (0.47) GRM4P2RX3ALDH1A1KDM4EHPGD
SCHEMBL28053931 0.80 NFE2L2 (0.55) GRM4ALDH1A1KDM4ERAB9AMEN1
SCHEMBL28053952 0.80 CYP11B1 (0.56) GRM4KDM4ERAB9AMEN1KMT2A
SCHEMBL20144415 0.79 BCHE (0.44) PTGS1PTGS2
SCHEMBL28053932 0.77 RELA (0.58) ALDH1A1KDM4EHPGDRAB9ANPC1
SCHEMBL6323560 0.77 MEN1 (0.54) GRM4ALDH1A1KDM4EHPGDRAB9A
SCHEMBL6323554 0.77 MEN1 (0.54) GRM4ALDH1A1KDM4EHPGDRAB9A
SCHEMBL10719653 0.73 GRM4 (0.50) GRM4P2RX3ALDH1A1KDM4EHPGD
SCHEMBL22721962 0.73 CHAT (0.45) ALDH1A1KDM4EHPGDRAB9AMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-103864768-B Ligustrazine stilbenoids derivatives and preparation method thereof and application GUANGXI NORMAL UNIVERSITY (CN) 2016-04-06 CN disclosed