SCHEMBL28053802

SCHEMBL28053802

Cc1nc(C)c(C=Cc2ccncc2)nc1C

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALOX5 P09917 1/20 0.47
MAPT P10636 6/20 0.46
NPC1 O15118 4/20 0.46
SMN1; SMN2 Q16637 3/20 0.46
RAB9A P51151 3/20 0.46
CYP1A2 P05177 2/20 0.46
HPGD P15428 2/20 0.46
KDM4E B2RXH2 2/20 0.46
MEN1 O00255 1/20 0.46
ALOX15 P16050 1/20 0.46
CASP1 P29466 1/20 0.46
HBB P68871 1/20 0.46
KMT2A Q03164 1/20 0.46
CYP3A4 P08684 1/20 0.46
CYP2D6 P10635 1/20 0.46
CYP2C9 P11712 1/20 0.46
CYP2C19 P33261 1/20 0.46
CYP1A1 P04798 2/20 0.43
CYP1B1 Q16678 2/20 0.43
ALDH1A1 P00352 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28053799 0.82 GRM4 (0.56) ALOX5MAPTNPC1SMN1; SMN2RAB9A
SCHEMBL28053931 0.78 NFE2L2 (0.55) ALOX5MAPTNPC1RAB9AKDM4E
SCHEMBL9000448 0.78 MAPT (0.50) ALOX5MAPTNPC1SMN1; SMN2RAB9A
SCHEMBL9000449 0.78 MAPT (0.50) ALOX5MAPTNPC1SMN1; SMN2RAB9A
SCHEMBL28053952 0.78 CYP11B1 (0.56) ALOX5MAPTNPC1RAB9AKDM4E
SCHEMBL20144415 0.78 BCHE (0.44) TXNRD1TXNRD3TXNRD2BCHEACHE
SCHEMBL28053932 0.76 RELA (0.58) ALOX5MAPTNPC1SMN1; SMN2RAB9A
SCHEMBL107198 0.75 MAPT (0.61) ALOX5MAPTNPC1SMN1; SMN2RAB9A
SCHEMBL138489 0.75 MAPT (0.61) ALOX5MAPTNPC1SMN1; SMN2RAB9A
SCHEMBL9966009 0.72 MAPT (0.65) ALOX5MAPTNPC1SMN1; SMN2RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-103864768-B Ligustrazine stilbenoids derivatives and preparation method thereof and application GUANGXI NORMAL UNIVERSITY (CN) 2016-04-06 CN disclosed