SCHEMBL28056343

SCHEMBL28056343

O=C(O)Cc1ccnnc1-c1ccccc1Cl

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NR4A2 P43354 2/20 0.45
KDM4E B2RXH2 1/20 0.45
ALDH1A1 P00352 1/20 0.45
RXFP1 Q9HBX9 1/20 0.45
CXCL8 P10145 3/20 0.43
CYP2C19 P33261 1/20 0.41
NR1H4 Q96RI1 2/20 0.41
TTR P02766 2/20 0.41
AKR1B10 O60218 1/20 0.41
UGT1A9 O60656 1/20 0.41
TRPA1 O75762 1/20 0.41
ABCB11 O95342 1/20 0.41
MT-CO2 P00403 1/20 0.41
ALB P02768 1/20 0.41
UGT1A6 P19224 1/20 0.41
UGT1A1 P22309 1/20 0.41
PTGS1 P23219 1/20 0.41
CXCR1 P25024 1/20 0.41
ADRA1A P35348 1/20 0.41
PTGS2 P35354 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28056298 0.84 AKR1B1 (0.51) KDM4EALDH1A1TTRAKR1B1HSD17B10
SCHEMBL28056374 0.77 ALDH1A1 (0.47) KDM4EALDH1A1HSD17B10KMT2A
SCHEMBL9890641 0.74 CXCL8 (0.57) NR4A2KDM4EALDH1A1RXFP1CXCL8
SCHEMBL6545903 0.73 ALDH1A1 (0.47) KDM4EALDH1A1DPP4HSD17B10KMT2A
SCHEMBL11258381 0.72 TDP1 (0.48) NR4A2KDM4EALDH1A1RXFP1CXCL8
SCHEMBL194831 0.69 CXCL8 (0.65) CXCL8NR1H4TTRAKR1B10UGT1A9
SCHEMBL29933245 0.69 CXCL8 (0.65) CXCL8NR1H4TTRAKR1B10UGT1A9
SCHEMBL5266212 0.69 DPP4 (0.44) NR4A2KDM4EALDH1A1ADRA1ADPP4
SCHEMBL34471968 0.69 ALPL (0.42) KDM4EALDH1A1HSD17B10KMT2AMAPT
SCHEMBL8396823 0.69 RXFP1 (0.49) NR4A2KDM4EALDH1A1RXFP1CXCL8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105503877-A Imidazopyridazine compound and application thereof HUTCHISON MEDIPHARMA LTD 2016-04-20 CN disclosed