SCHEMBL28056859

SCHEMBL28056859

CCOC(=O)c1ccc(C(=O)N2CCC3CC=CC=C3C2)cc1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
FDFT1 P37268 1/20 0.47
ALDH1A1 P00352 4/20 0.44
TDP1 Q9NUW8 1/20 0.44
SMN1; SMN2 Q16637 2/20 0.42
KMT2A Q03164 2/20 0.42
HTT P42858 2/20 0.42
LMNA P02545 1/20 0.42
RAB9A P51151 4/20 0.40
NPC1 O15118 2/20 0.40
MEN1 O00255 1/20 0.40
GAA P10253 1/20 0.40
TSHR P16473 1/20 0.40
CA12 O43570 1/20 0.40
CA1 P00915 1/20 0.40
CA2 P00918 1/20 0.40
ESR1 P03372 1/20 0.40
CA7 P43166 1/20 0.40
CA9 Q16790 1/20 0.40
ESR2 Q92731 1/20 0.40
CA14 Q9ULX7 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28949869 0.87 EPHX1 (0.43) ALDH1A1KMT2AHTTMEN1GAA
SCHEMBL28056844 0.85 LMNA (0.45) ALDH1A1TDP1SMN1; SMN2KMT2ALMNA
SCHEMBL28056837 0.84 ABL1 (0.40) KMT2ALMNAMEN1GAA
SCHEMBL28056726 0.82 NPC1 (0.41) KMT2ALMNARAB9ANPC1MEN1
SCHEMBL28056784 0.81 PARP10 (0.46) ALDH1A1TDP1SMN1; SMN2RAB9ANPC1
SCHEMBL10922111 0.75 QDPR (0.40) ALDH1A1
SCHEMBL28166840 0.72 PDE4B (0.32) SMN1; SMN2CA12CA1CA2CA7
SCHEMBL3033970 0.70 FDFT1 (0.55) FDFT1ALDH1A1TDP1SMN1; SMN2HTT
SCHEMBL3040729 0.69 FDFT1 (0.53) FDFT1ALDH1A1TDP1SMN1; SMN2KMT2A
SCHEMBL28056773 0.69 MEN1 (0.72) ALDH1A1KMT2AHTTLMNARAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-103732589-B Can be used as the sulphonamide of the replacement of anti-apoptotic BCL inhibitor BRISTOL-MYERS SQUIBB CO. (US) 2016-03-30 CN disclosed