SCHEMBL28060419

SCHEMBL28060419

CC(C)(C)C(=O)ON1CCC(C(=O)NC2CC2)CC1

nearest known ligand 0.44

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
MAPK1 P28482 2/20 0.44
GAA P10253 2/20 0.43
ALDH1A1 P00352 5/20 0.42
RAB9A P51151 2/20 0.42
NPC1 O15118 1/20 0.42
EPHX2 P34913 6/20 0.41
MEN1 O00255 1/20 0.41
KMT2A Q03164 1/20 0.41
L3MBTL1 Q9Y468 2/20 0.41
LMNA P02545 2/20 0.41
TSHR P16473 1/20 0.40
CYP3A4 P08684 1/20 0.40
CYP2C9 P11712 1/20 0.40
CYP2C19 P33261 1/20 0.40
TDP1 Q9NUW8 1/20 0.40
POLB P06746 1/20 0.40
KDM4E B2RXH2 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27968794 0.82 PTPN2 (0.37) GAAALDH1A1RAB9ANPC1KMT2A
SCHEMBL16992001 0.80 MAPK1 (0.49) MAPK1GAAALDH1A1RAB9ANPC1
SCHEMBL27987722 0.80 L3MBTL1 (0.39) MAPK1ALDH1A1RAB9ANPC1EPHX2
SCHEMBL28060472 0.79 HTT (0.45) MAPK1GAAALDH1A1EPHX2LMNA
SCHEMBL28060475 0.79 CTSK (0.42) GAAALDH1A1EPHX2LMNACYP2C9
SCHEMBL1437590 0.78 EPHX2 (0.49) MAPK1GAAALDH1A1EPHX2L3MBTL1
SCHEMBL28064466 0.78 SMN1; SMN2 (0.54) GAAALDH1A1RAB9ANPC1MEN1
SCHEMBL27643661 0.78 HPGD (0.36) ALDH1A1MEN1KMT2ALMNATSHR
SCHEMBL27566300 0.78 HPGD (0.36) ALDH1A1MEN1KMT2ALMNATSHR
SCHEMBL1514783 0.77 EPHX1 (0.64) MAPK1ALDH1A1RAB9ANPC1EPHX2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109851610-A Azabicyclo compound as muscarine M1 and/or M4 receptor stimulating agent 赫普泰雅治疗有限公司 2019-06-07 CN disclosed
CN-106458986-B Bicyclic aza compounds as muscarinic M1 and/or M4 receptor agonists 赫普泰雅治疗有限公司 2019-01-04 CN disclosed
CN-106458986-A Bicyclic aza compounds as muscarinic M1 and/or M4 receptor agonists 赫普泰雅治疗有限公司 2017-02-22 CN disclosed
CN-105399698-A Aromatic heterocyclic derivatives and applications of aromatic heterocyclic derivatives in medicines GUANGDONG HEC PHARMACEUTICAL 2016-03-16 CN disclosed