SCHEMBL28061498

SCHEMBL28061498

NNC(=O)N(N)c1ncc(F)cc1F

nearest known ligand 0.34

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
HTT P42858 1/20 0.34
MEN1 O00255 1/20 0.32
CYP1A2 P05177 1/20 0.32
CYP3A4 P08684 1/20 0.32
GAA P10253 1/20 0.32
CYP2C19 P33261 1/20 0.32
KMT2A Q03164 1/20 0.32
ALPL P05186 1/20 0.32
AGBL2 Q5U5Z8 1/20 0.31
CDK8 P49336 1/20 0.31
GSK3A P49840 1/20 0.31
GSK3B P49841 1/20 0.31
CDK9 P50750 1/20 0.31
CDK5 Q00535 1/20 0.31
DYRK1B Q9Y463 1/20 0.31
BACE1 P56817 2/20 0.31
PIK3C3 Q8NEB9 1/20 0.30
SSTR4 P31391 1/20 0.30
LMNA P02545 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28453095 0.80 AGBL2 (0.39) HTTAGBL2PIK3C3SSTR4
SCHEMBL107626 0.69 BACE1 (0.42) HTTGAAALPLAGBL2BACE1
SCHEMBL29570161 0.67 CES2 (0.39) HTTGAAALPLLMNA
SCHEMBL28058122 0.67 GAA (0.38) HTTMEN1GAAKMT2ABACE1
SCHEMBL27861418 0.67 TSHR (0.34) MEN1CYP3A4GAAKMT2ACDK8
SCHEMBL27812260 0.66 GRM5 (0.31) MEN1CYP1A2CYP3A4GAACYP2C19
SCHEMBL27819606 0.66 GRM5 (0.39) MEN1CYP1A2CYP3A4GAACYP2C19
SCHEMBL27840502 0.66 P2RX7 (0.34)
SCHEMBL9363725 0.65 P2RX7 (0.32)
SCHEMBL9037566 0.65 ALDH1A1 (0.39) MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-103936717-B A kind of delafloxacin intermediate and preparation method thereof 上海医药工业研究院 2016-08-10 CN disclosed