SCHEMBL28062036

SCHEMBL28062036

O=C(CS)CCc1ccccc1

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KEAP1 Q14145 1/20 0.61
ALDH1A1 P00352 2/20 0.57
FFAR1 O14842 2/20 0.57
TDP1 Q9NUW8 2/20 0.55
TRPA1 O75762 2/20 0.55
L3MBTL1 Q9Y468 1/20 0.55
HDAC2 Q92769 3/20 0.53
HDAC8 Q9BY41 3/20 0.53
HDAC6 Q9UBN7 3/20 0.53
HDAC1 Q13547 3/20 0.52
HDAC3 O15379 2/20 0.52
HDAC4 P56524 2/20 0.52
HDAC7 Q8WUI4 2/20 0.52
HDAC10 Q969S8 2/20 0.52
HDAC11 Q96DB2 2/20 0.52
HDAC9 Q9UKV0 2/20 0.52
HDAC5 Q9UQL6 2/20 0.52
MAPK1 P28482 1/20 0.52
ADRA1A P35348 1/20 0.52
SLC6A3 Q01959 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL497371 0.86 KEAP1 (0.73) KEAP1ALDH1A1FFAR1TDP1TRPA1
SCHEMBL11275710 0.86 MAPT (0.69) TDP1TRPA1HDAC2HDAC8HDAC6
SCHEMBL156142 0.84 KEAP1 (0.64) KEAP1ALDH1A1FFAR1TDP1TRPA1
SCHEMBL107423 0.84 KEAP1 (0.70) KEAP1ALDH1A1FFAR1TDP1TRPA1
SCHEMBL712597 0.84 KEAP1 (0.70) KEAP1ALDH1A1FFAR1TDP1TRPA1
SCHEMBL19561359 0.83 HDAC1 (0.69) KEAP1ALDH1A1FFAR1TDP1TRPA1
SCHEMBL5598977 0.82 KEAP1 (0.67) KEAP1ALDH1A1FFAR1TDP1TRPA1
SCHEMBL19625551 0.81 MAPT (0.68) KEAP1ALDH1A1FFAR1TDP1TRPA1
SCHEMBL452362 0.80 TDP1 (0.79) KEAP1ALDH1A1FFAR1TDP1TRPA1
SCHEMBL27474155 0.80 KEAP1 (0.64) KEAP1ALDH1A1FFAR1TDP1TRPA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-104136433-B Antiviral compounds with a heterotricyclic moiety LUPIN LTD. (IN) 2016-05-04 CN disclosed