SCHEMBL28062609

SCHEMBL28062609

C#CCC(C(=O)c1cc(F)c(F)cc1F)N(C(=O)O)C(C)(C)C

nearest known ligand 0.31

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
POLB P06746 1/20 0.31
APEX1 P27695 1/20 0.31
MAOA P21397 1/20 0.30
MAOB P27338 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17102154 0.86 CES2 (0.40)
SCHEMBL28062336 0.73 MAOA (0.32) MAOAMAOB
SCHEMBL28062335 0.73 MAOA (0.32) MAOAMAOB
SCHEMBL18760099 0.69
SCHEMBL17865487 0.67 CES2 (0.40)
SCHEMBL28037292 0.66 CES2 (0.36) MAOAMAOB
SCHEMBL28037291 0.66 CES2 (0.36) MAOAMAOB
SCHEMBL17373217 0.66
SCHEMBL28044516 0.66
SCHEMBL16993854 0.64 GRIK1 (0.33)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105518008-B Amino pyrans ring derivatives and combinations thereof and application 海思科医药集团股份有限公司 2018-03-27 CN disclosed
CN-105531277-B Pyrrolo-imidazole ring derivatives and their use in medicine 四川海思科制药有限公司 2018-03-02 CN disclosed
CN-105531277-A Pyrrolo-imidazole ring derivatives and their use in medicine SICHUAN HAISCO PHARMACEUTICAL CO LTD 2016-04-27 CN disclosed
CN-105518008-A Amino pyranoid ring derivative and composition and use thereof SICHUAN HAISCO PHARMACEUTICAL CO LTD 2016-04-20 CN disclosed