SCHEMBL28067939

SCHEMBL28067939

Fc1ccc2c(c1)C=NC2

nearest known ligand 0.38

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
HTR5A P47898 4/20 0.38
ADRA2A P08913 2/20 0.35
ADRA2B P18089 1/20 0.32
ADRA2C P18825 1/20 0.32
SLC6A4 P31645 1/20 0.32
ACHE P22303 1/20 0.32
PARP1 P09874 1/20 0.32
PARP10 Q53GL7 1/20 0.32
KDM4E B2RXH2 1/20 0.31
ROCK1 Q13464 1/20 0.31
NOS3 P29474 1/20 0.31
KDM1A O60341 1/20 0.31
KMT2A Q03164 1/20 0.31
HTR2A P28223 1/20 0.30
HTR2C P28335 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9572969 0.79 ADRA2A (0.39) HTR5AADRA2AADRA2BADRA2CSLC6A4
SCHEMBL29458622 0.79 ADRA2A (0.39) HTR5AADRA2AADRA2BADRA2CSLC6A4
Hydrochloric Acid SCHEMBL11658196 0.78 ADRA2A (0.38) HTR5AADRA2APARP1PARP10KDM1A
SCHEMBL18023177 0.74 MAPT (0.35) ADRA2ASLC6A4ACHEKDM4EKMT2A
SCHEMBL2965836 0.74 TRPA1 (0.47) ADRA2AADRA2BADRA2CPARP1PARP10
SCHEMBL7934799 0.74 HTR5A (0.38) HTR5AADRA2AACHEPARP1PARP10
SCHEMBL11795867 0.69 HTR7 (0.35) HTR2AHTR2C
SCHEMBL15528512 0.69 TRPA1 (0.51) KDM1A
SCHEMBL8824570 0.67 HTR5A (0.33) HTR5AADRA2AADRA2BADRA2CACHE
SCHEMBL29517242 0.67

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-103732596-B Pyrrolopyrimidine derivatives NOVARTIS AG (CH) 2016-06-01 CN disclosed