Guanosine

Guanosine

SCHEMBL28068227

Nc1nc2c(ncn2[C@@H]2O[C@H](CO)[C@@H](O)[C@H]2O)c(=O)[nH]1.O=CC(O)C(O)C(O)CO.O=P(O)(O)O

nearest known ligand 0.58

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Known targets — ChEMBL curated mechanism

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

The experimentally established mechanism targets of Guanosine. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
NT5E P21589 1/20 0.58
HPGD P15428 1/20 0.56
TGM2 P21980 1/20 0.54
HINT1 P49773 1/20 0.52
IMPDH2 P12268 3/20 0.51
KRAS P01116 5/20 0.51
GSK3A P49840 2/20 0.49
RPS6KA3 P51812 2/20 0.49
MAPK14 Q16539 2/20 0.49
FUT5 Q11128 1/20 0.49
IMPDH1 P20839 1/20 0.49
PNP P00491 1/20 0.49
PAX8 Q06710 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Guanosine SCHEMBL19810340 0.97 HPGD (0.59) NT5EHPGDTGM2HINT1GSK3A
Guanosine SCHEMBL3977221 0.97 HPGD (0.59) NT5EHPGDTGM2HINT1GSK3A
Guanosine SCHEMBL19810339 0.97 HPGD (0.59) NT5EHPGDTGM2HINT1GSK3A
Guanosine SCHEMBL28166235 0.96 HPGD (0.58) NT5EHPGDTGM2HINT1GSK3A
Guanosine SCHEMBL28048641 0.95 TGM2 (0.57) NT5EHPGDTGM2HINT1IMPDH2
Guanosine SCHEMBL11066196 0.94 HPGD (0.58) NT5EHPGDTGM2HINT1GSK3A
Guanosine SCHEMBL22498410 0.94 HPGD (0.58) NT5EHPGDTGM2HINT1GSK3A
Guanosine SCHEMBL22498408 0.94 HPGD (0.58) NT5EHPGDTGM2HINT1GSK3A
E626 SCHEMBL27748771 0.91 NT5E (0.66) NT5ETGM2HINT1IMPDH2KRAS
Guanosine SCHEMBL22498413 0.91 HPGD (0.54) NT5EHPGDTGM2HINT1GSK3A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105524609-B A kind of fluorescence probe GH and its preparation and application 中国科学院大连化学物理研究所 2017-09-22 CN claimed
CN-105524609-A Fluorescent probe GH and preparation method and application thereof DALIAN INST CHEMICAL PHYSICS CAS 2016-04-27 CN claimed
CN-105524609-B A kind of fluorescence probe GH and its preparation and application 中国科学院大连化学物理研究所 2017-09-22 CN disclosed
CN-105524609-B A kind of fluorescence probe GH and its preparation and application 中国科学院大连化学物理研究所 2017-09-22 CN disclosed
CN-105524609-A Fluorescent probe GH and preparation method and application thereof DALIAN INST CHEMICAL PHYSICS CAS 2016-04-27 CN disclosed