SCHEMBL28068682

SCHEMBL28068682

CC(=O)Oc1ccc(Cl)c(C#N)c1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MRGPRX4 Q96LA9 1/20 0.48
PLA2G7 Q13093 1/20 0.45
LMNA P02545 3/20 0.43
KDM4E B2RXH2 3/20 0.42
VCAM1 P19320 1/20 0.42
CYP3A4 P08684 2/20 0.42
AR P10275 2/20 0.42
ACHE P22303 2/20 0.41
CUL4A Q13619 1/20 0.41
ACACB O00763 1/20 0.40
GRM4 Q14833 1/20 0.40
POLB P06746 2/20 0.40
MAPT P10636 2/20 0.40
CA12 O43570 1/20 0.40
GLA P06280 1/20 0.40
GAA P10253 1/20 0.40
CA9 Q16790 1/20 0.40
TDP1 Q9NUW8 1/20 0.40
PKM P14618 1/20 0.40
MEN1 O00255 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8071507 0.87 AR (0.54) MRGPRX4LMNAKDM4ECYP3A4AR
SCHEMBL5263668 0.81 ACHE (0.54) LMNAKDM4ECYP3A4ARACHE
SCHEMBL5630201 0.81 CYP3A4 (0.47) LMNAKDM4ECYP3A4ARACHE
SCHEMBL28397412 0.80 LMNA (0.43) LMNAKDM4ECYP3A4ARACHE
SCHEMBL21728056 0.80 LMNA (0.43) LMNAKDM4ECYP3A4ARACHE
SCHEMBL473532 0.78 LMNA (0.52) LMNAKDM4ECYP3A4ACHEPOLB
SCHEMBL27935121 0.78 KDM4E (0.56) LMNAKDM4ECYP3A4ARACHE
SCHEMBL21719017 0.78 CYP3A4 (0.44) LMNAKDM4ECYP3A4ARACHE
SCHEMBL10662281 0.77 MEN1 (0.45) MRGPRX4KDM4EVCAM1ARPOLB
SCHEMBL2733341 0.77 LMNA (0.43) LMNAKDM4ECYP3A4ARACHE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-103687860-B As P2X7Heterocyclic amide derivatives of receptor antagonists 埃科特莱茵药品有限公司 2016-06-08 CN disclosed