SCHEMBL28074550

SCHEMBL28074550

Cc1cccn1S(=O)(=O)c1ccc(F)cc1

nearest known ligand 0.49

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
RAPGEF4 Q8WZA2 3/20 0.49
ALDH3A1 P30838 2/20 0.46
PKM P14618 1/20 0.46
PPME1 Q9Y570 1/20 0.45
TSHR P16473 2/20 0.45
MEN1 O00255 3/20 0.44
KMT2A Q03164 3/20 0.44
ALDH1A1 P00352 2/20 0.44
LMNA P02545 2/20 0.44
MAPK1 P28482 1/20 0.44
HTT P42858 1/20 0.44
MMP2 P08253 1/20 0.43
CA1 P00915 1/20 0.42
CA2 P00918 1/20 0.42
GAA P10253 1/20 0.41
NPSR1 Q6W5P4 1/20 0.41
HTR6 P50406 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3834757 0.85 RAPGEF4 (0.65) RAPGEF4ALDH3A1PKMALDH1A1HTT
SCHEMBL1599348 0.83 HTR6 (0.50) RAPGEF4PPME1TSHRMEN1KMT2A
SCHEMBL11932215 0.79 RAPGEF4 (0.66) RAPGEF4PKMTSHRMEN1KMT2A
SCHEMBL28458237 0.78 RAPGEF4 (0.52) RAPGEF4ALDH3A1PKMLMNAHTT
SCHEMBL3968075 0.76 PPME1 (0.55) RAPGEF4ALDH3A1PKMPPME1MEN1
SCHEMBL30427800 0.76 HTR6 (0.52) ALDH3A1PKMPPME1TSHRMEN1
SCHEMBL5535689 0.75 RAPGEF4 (0.61) RAPGEF4ALDH3A1PKMALDH1A1HTT
SCHEMBL13381696 0.72 KDM4E (0.53) ALDH3A1TSHRKMT2AALDH1A1HTT
SCHEMBL30041811 0.70 HTR6 (0.53) RAPGEF4ALDH3A1KMT2AALDH1A1LMNA
SCHEMBL3967709 0.69 HTR6 (0.75) RAPGEF4ALDH3A1PKMTSHRMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105612153-B Substituted heterocyclic sulfonamide compound as TRPA1 conditioning agents 豪夫迈·罗氏有限公司 2018-09-14 CN disclosed
CN-105612153-A Substituted sulfonamide compounds as TRPA1 conditioner HOFFMANN LA ROCHE 2016-05-25 CN disclosed