SCHEMBL28074643

SCHEMBL28074643

NC(=O)c1cn(-c2cnc(C(F)(F)F)nc2)nc1O

nearest known ligand 0.41

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 5/20 0.41
SCN9A Q15858 1/20 0.34
PARP2 Q9UGN5 2/20 0.34
PARP3 Q9Y6F1 2/20 0.34
CA12 O43570 4/20 0.34
CA1 P00915 4/20 0.34
CA2 P00918 4/20 0.34
CA9 Q16790 4/20 0.34
TRPA1 O75762 5/20 0.33
KMT2A Q03164 2/20 0.33
FGFR1 P11362 1/20 0.33
HDAC11 Q96DB2 1/20 0.33
ALDH1A1 P00352 2/20 0.33
KDM4E B2RXH2 1/20 0.33
PKM P14618 1/20 0.33
L3MBTL1 Q9Y468 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16635561 0.81 TRPA1 (0.43) PARP1SCN9ACA12CA1CA2
SCHEMBL28210218 0.73 PARP1 (0.59) PARP1PARP2PARP3CA12CA1
SCHEMBL17973850 0.70 TRPA1 (0.43) TRPA1KMT2AFGFR1HDAC11ALDH1A1
SCHEMBL16635488 0.70 TRPA1 (0.43) TRPA1KMT2AHDAC11ALDH1A1L3MBTL1
SCHEMBL24487886 0.69 NFKB1 (0.51) CA12CA9KMT2AALDH1A1KDM4E
SCHEMBL2871260 0.68 NNMT (0.45) KMT2AKDM4EL3MBTL1
SCHEMBL19795577 0.68 JUN (0.50) ALDH1A1KDM4E
SCHEMBL16635272 0.66 NFKB1 (0.48) CA12CA9TRPA1ALDH1A1KDM4E
SCHEMBL19807437 0.66 TRPA1 (0.52) TRPA1FGFR1ALDH1A1KDM4E
SCHEMBL14307992 0.66 PARP1 (0.54) PARP1SCN9APARP2PARP3CA12

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105612153-A Substituted sulfonamide compounds as TRPA1 conditioner HOFFMANN LA ROCHE 2016-05-25 CN disclosed