SCHEMBL28076706

SCHEMBL28076706

COc1cc(CC2CCN(CCC(O)c3ccccc3Cl)CC2)c(N)cc1C(N)=O

nearest known ligand 0.43

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
ACHE P22303 6/20 0.43
DRD4 P21917 3/20 0.43
DRD2 P14416 2/20 0.43
DRD3 P35462 2/20 0.43
HTR4 Q13639 8/20 0.43
MEN1 O00255 2/20 0.43
KMT2A Q03164 2/20 0.43
ALDH1A1 P00352 1/20 0.42
CYP2D6 P10635 1/20 0.42
CYP2C9 P11712 1/20 0.42
TSHR P16473 1/20 0.42
KCNH2 Q12809 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28816405 0.97 ACHE (0.45) ACHEDRD4DRD2DRD3HTR4
SCHEMBL27997559 0.90 ACHE (0.44) ACHEDRD4DRD2DRD3HTR4
SCHEMBL28076576 0.90 GRIN2B (0.41) ACHEDRD4DRD2DRD3HTR4
SCHEMBL27997525 0.90 MEN1 (0.43) ACHEDRD4DRD2DRD3HTR4
SCHEMBL27997565 0.88 ACHE (0.46) ACHEDRD4DRD2DRD3HTR4
SCHEMBL27997756 0.86 HTR4 (0.42) ACHEDRD4DRD2DRD3HTR4
SCHEMBL28076538 0.86 HTR4 (0.44) ACHEDRD4HTR4MEN1KMT2A
SCHEMBL28076529 0.86 CCR5 (0.41) ACHEDRD4DRD2DRD3HTR4
SCHEMBL28076702 0.84 MCHR1 (0.49) ACHEDRD4DRD2DRD3MEN1
SCHEMBL27997728 0.83 HTR4 (0.46) ACHEDRD4HTR4MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-103980184-B Piperidine compounds, medical composition and its use containing this compound 爱思开生物制药株式会社 2016-08-24 CN claimed