SCHEMBL28076795

SCHEMBL28076795

COc1ccc(CC2CCN(CCC(O)c3cccc(F)c3)CC2)c(N)c1

nearest known ligand 0.50

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
HTR1A P08908 7/20 0.46
SLC6A4 P31645 6/20 0.46
GRIN2B Q13224 3/20 0.44
RYR2 Q92736 1/20 0.43
MCHR1 Q99705 1/20 0.43
MAPT P10636 1/20 0.43
ALOX12 P18054 1/20 0.43
L3MBTL1 Q9Y468 1/20 0.43
MEN1 O00255 1/20 0.42
KMT2A Q03164 1/20 0.42
CCR3 P51677 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28076884 0.90 SLC6A4 (0.52) HTR1ASLC6A4GRIN2BRYR2CCR3
SCHEMBL28076765 0.89 HTR1A (0.52) HTR1ASLC6A4RYR2MCHR1MAPT
SCHEMBL28076801 0.84 HTR1A (0.52) HTR1ASLC6A4GRIN2BRYR2MAPT
SCHEMBL28076771 0.84 HTR1A (0.52) HTR1ASLC6A4GRIN2BRYR2
SCHEMBL27997732 0.83 SLC6A4 (0.41) SLC6A4GRIN2BMCHR1MEN1KMT2A
SCHEMBL28076769 0.82 HTR1A (0.52) HTR1ASLC6A4RYR2MAPTALOX12
SCHEMBL28076798 0.80 HTR1A (0.55) HTR1ASLC6A4RYR2CCR3
SCHEMBL28076620 0.78 HTR1A (0.46) HTR1ASLC6A4GRIN2BRYR2MAPT
SCHEMBL28076611 0.75 MAPT (0.48) HTR1ASLC6A4GRIN2BRYR2MAPT
SCHEMBL28830757 0.74 TSHR (0.60) MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105646331-B Piperidine compounds, the medical composition and its use containing the compound 爱思开生物制药株式会社 2018-07-03 CN disclosed
CN-103980184-B Piperidine compounds, medical composition and its use containing this compound 爱思开生物制药株式会社 2016-08-24 CN disclosed