SCHEMBL28076771

SCHEMBL28076771

COc1ccc(CC2CCN(CCC(O)c3ccc(Cl)cc3)CC2)c(N)c1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR1A P08908 11/20 0.52
SLC6A4 P31645 9/20 0.52
GRIN1 Q05586 2/20 0.46
GRIN2B Q13224 2/20 0.46
GRIN2D O15399 1/20 0.46
GRIN3B O60391 1/20 0.46
ADRA1D P25100 1/20 0.46
ADRA1A P35348 1/20 0.46
ADRA1B P35368 1/20 0.46
GRIN2A Q12879 1/20 0.46
GRIN2C Q14957 1/20 0.46
GRIN3A Q8TCU5 1/20 0.46
RYR2 Q92736 1/20 0.45
DRD4 P21917 3/20 0.45
GMNN O75496 1/20 0.44
TP53 P04637 1/20 0.44
CYP3A4 P08684 1/20 0.44
ALOX15 P16050 1/20 0.44
TSHR P16473 1/20 0.44
NFKB1 P19838 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28076884 0.90 SLC6A4 (0.52) HTR1ASLC6A4GRIN1GRIN2BGRIN2D
SCHEMBL28076765 0.90 HTR1A (0.52) HTR1ASLC6A4RYR2
SCHEMBL28076769 0.85 HTR1A (0.52) HTR1ASLC6A4RYR2
SCHEMBL28076795 0.84 HTR1A (0.46) HTR1ASLC6A4GRIN2BRYR2
SCHEMBL27997728 0.82 HTR4 (0.46) GRIN1GRIN2BGRIN2DGRIN3BADRA1D
SCHEMBL28076538 0.82 HTR4 (0.44) GRIN1GRIN2BGRIN2DGRIN3BADRA1D
SCHEMBL28076611 0.81 MAPT (0.48) HTR1ASLC6A4GRIN1GRIN2BRYR2
SCHEMBL28076801 0.81 HTR1A (0.52) HTR1ASLC6A4GRIN2BRYR2
SCHEMBL28830809 0.80 DRD4 (0.62) DRD4
SCHEMBL28076620 0.78 HTR1A (0.46) HTR1ASLC6A4GRIN1GRIN2BADRA1D

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-103980184-B Piperidine compounds, medical composition and its use containing this compound 爱思开生物制药株式会社 2016-08-24 CN disclosed