SCHEMBL28830757

SCHEMBL28830757

COc1ccc(CC2CCN(CC(O)COc3ccc(F)cc3)CC2)c(N)c1

nearest known ligand 0.60

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
TSHR P16473 1/20 0.60
DRD4 P21917 5/20 0.59
CACNA1G O43497 1/20 0.57
GAA P10253 1/20 0.56
MEN1 O00255 3/20 0.55
KMT2A Q03164 3/20 0.55
CYP2D6 P10635 3/20 0.53
KDM4E B2RXH2 1/20 0.50
POLB P06746 1/20 0.50
USP2 O75604 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28830809 0.90 DRD4 (0.62) DRD4CACNA1GGAAMEN1KMT2A
SCHEMBL28076585 0.85 DRD4 (0.58) DRD4GAAMEN1KMT2AUSP2
SCHEMBL28076710 0.84 TSHR (0.52) TSHRDRD4CACNA1GGAAMEN1
SCHEMBL27997731 0.84 TSHR (0.52) TSHRDRD4CACNA1GGAAMEN1
SCHEMBL28076582 0.82 CYP2D6 (0.55) DRD4GAACYP2D6
SCHEMBL28076798 0.81 HTR1A (0.55)
SCHEMBL28076624 0.80 HTR1A (0.52) DRD4GAAMEN1KMT2APOLB
SCHEMBL28076884 0.80 SLC6A4 (0.52) TSHR
SCHEMBL28076704 0.79 GAA (0.56) DRD4GAAMEN1KMT2ACYP2D6
SCHEMBL28076620 0.78 HTR1A (0.46) TSHRDRD4GAAMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-103980184-B Piperidine compounds, medical composition and its use containing this compound 爱思开生物制药株式会社 2016-08-24 CN disclosed