SCHEMBL28077873

SCHEMBL28077873

CC(C)(C)C(=O)ON1CCC(CC#N)(c2ccc(Cl)cc2)CC1

nearest known ligand 0.39

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 5/20 0.39
OPRM1 P35372 3/20 0.38
CCR1 P32246 3/20 0.37
P2RX7 Q99572 1/20 0.36
EPHX2 P34913 1/20 0.35
HSD11B1 P28845 1/20 0.35
NPC1 O15118 1/20 0.34
CYP1A2 P05177 1/20 0.34
CYP2C9 P11712 1/20 0.34
CYP2C19 P33261 1/20 0.34
KMT2A Q03164 1/20 0.34
OPRL1 P41146 1/20 0.34
PDE4A P27815 1/20 0.34
PDE4B Q07343 1/20 0.34
PDE4C Q08493 1/20 0.34
PDE4D Q08499 1/20 0.34
CYP3A4 P08684 1/20 0.34
CNR1 P21554 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28755147 0.89 ALDH1A1 (0.35) HSD11B1NPC1KMT2APDE4APDE4B
SCHEMBL28077607 0.89 EPHX2 (0.45) DRD2OPRM1CCR1P2RX7EPHX2
SCHEMBL27640160 0.87 SLC6A4 (0.38) OPRM1CCR1HSD11B1PDE4APDE4B
SCHEMBL27621503 0.87 CCR5 (0.39) CCR1HSD11B1
SCHEMBL27640204 0.86 HSD11B1 (0.34) HSD11B1KMT2APDE4APDE4BPDE4C
SCHEMBL27640138 0.85 JAK2 (0.41) OPRM1CCR1HSD11B1CYP2C9CYP2C19
SCHEMBL28831246 0.84 SLC6A4 (0.48) DRD2OPRM1P2RX7NPC1CYP1A2
SCHEMBL27640184 0.84 METAP2 (0.35) HSD11B1PDE4APDE4BPDE4CPDE4D
SCHEMBL28077735 0.83 OPRM1 (0.57) DRD2OPRM1CCR1PDE4APDE4B
SCHEMBL28077739 0.82 DRD2 (0.39) DRD2OPRM1CCR1P2RX7HSD11B1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105745209-A Triazolopyridine compounds, compositions, and methods of use thereof 豪夫迈·罗氏有限公司 2016-07-06 CN disclosed