SCHEMBL28077607

SCHEMBL28077607

CC(C)(C)C(=O)ON1CCC(CCC#N)(c2ccc(Cl)cc2)CC1

nearest known ligand 0.45

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
EPHX2 P34913 1/20 0.45
JAK2 O60674 1/20 0.38
JAK1 P23458 1/20 0.38
DRD2 P14416 5/20 0.38
HSD11B1 P28845 1/20 0.37
OPRM1 P35372 3/20 0.36
CCR1 P32246 3/20 0.36
CYP3A4 P08684 1/20 0.35
P2RX7 Q99572 1/20 0.35
NPC1 O15118 1/20 0.33
CYP1A2 P05177 1/20 0.33
CYP2C9 P11712 1/20 0.33
CYP2C19 P33261 1/20 0.33
KMT2A Q03164 1/20 0.33
OPRL1 P41146 1/20 0.33
CNR1 P21554 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28077873 0.89 DRD2 (0.39) EPHX2DRD2HSD11B1OPRM1CCR1
SCHEMBL28831246 0.82 SLC6A4 (0.48) DRD2OPRM1P2RX7NPC1CYP1A2
SCHEMBL16565440 0.82 MEN1 (0.47) EPHX2JAK2JAK1DRD2KMT2A
SCHEMBL28077735 0.81 OPRM1 (0.57) DRD2OPRM1CCR1
SCHEMBL16554233 0.81 EPHX2 (0.43) EPHX2JAK2JAK1DRD2HSD11B1
SCHEMBL28077739 0.81 DRD2 (0.39) DRD2HSD11B1OPRM1CCR1CYP3A4
SCHEMBL28077557 0.81 DRD2 (0.36) DRD2OPRM1CYP3A4P2RX7NPC1
SCHEMBL28077613 0.80 DRD2 (0.39) JAK2JAK1DRD2HSD11B1OPRM1
SCHEMBL28077553 0.79 DRD2 (0.50) DRD2P2RX7CNR1
SCHEMBL28755147 0.78 ALDH1A1 (0.35) JAK2JAK1HSD11B1NPC1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105745209-A Triazolopyridine compounds, compositions, and methods of use thereof 豪夫迈·罗氏有限公司 2016-07-06 CN disclosed