SCHEMBL28078633

SCHEMBL28078633

CC(C)c1c(N)ccc(C(N)=O)c1O

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ERN1 O75460 1/20 0.39
PARP1 P09874 1/20 0.37
IRAK4 Q9NWZ3 2/20 0.36
IKBKB O14920 1/20 0.36
ALDH1A1 P00352 3/20 0.35
MAPT P10636 2/20 0.35
KDM4E B2RXH2 1/20 0.35
HPGD P15428 1/20 0.35
TSHR P16473 1/20 0.35
HSD17B10 Q99714 1/20 0.35
KMT2A Q03164 2/20 0.33
MEN1 O00255 1/20 0.33
MAPK1 P28482 1/20 0.33
CDC7 O00311 1/20 0.33
GRK6 P43250 1/20 0.33
HTT P42858 2/20 0.32
GAA P10253 1/20 0.32
ALOX12 P18054 1/20 0.32
HIF1A Q16665 1/20 0.32
MMP2 P08253 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28423389 0.78 ALDH1A1 (0.40) ALDH1A1MAPTKDM4EHPGDTSHR
SCHEMBL2882576 0.78 IRAK4 (0.44) PARP1IRAK4ALDH1A1MAPTKDM4E
SCHEMBL3628076 0.76 IRAK4 (0.44) PARP1IRAK4IKBKBALDH1A1MAPT
SCHEMBL7216382 0.74 IKBKB (0.46) ERN1PARP1IKBKBALDH1A1MAPT
SCHEMBL16369793 0.74 IRAK4 (0.47) ERN1PARP1IRAK4ALDH1A1
SCHEMBL8980659 0.73 NNMT (0.38) ERN1IRAK4ALDH1A1MAPTKDM4E
SCHEMBL3424158 0.72 ERN1 (0.54) ERN1PARP1ALDH1A1MAPTKDM4E
SCHEMBL30211643 0.72 ERN1 (0.54) ERN1PARP1ALDH1A1MAPTKDM4E
SCHEMBL2922690 0.72 KDM4E (0.42) ALDH1A1MAPTKDM4EHPGDHSD17B10
SCHEMBL12316432 0.71 ERN1 (0.42) ERN1PARP1IKBKBALDH1A1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105793424-B Ascomycetes amides 亥姆霍兹感染研究中心有限公司 2021-02-19 CN disclosed
CN-105793424-A Ascomycetes amides 亥姆霍兹感染研究中心有限公司 2016-07-20 CN disclosed