SCHEMBL28079384

SCHEMBL28079384

Brc1cccc(N2CCNC2)c1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR7 P34969 5/20 0.50
ADRB1 P08588 4/20 0.50
HTR1A P08908 4/20 0.50
HTR3E A5X5Y0 4/20 0.50
HTR3B O95264 4/20 0.50
HTR3A P46098 4/20 0.50
HTR3D Q70Z44 4/20 0.50
HTR3C Q8WXA8 4/20 0.50
SIGMAR1 Q99720 4/20 0.50
HTR2C P28335 3/20 0.50
THRB P10828 2/20 0.50
HTR6 P50406 2/20 0.50
TP53 P04637 1/20 0.50
CYP1A2 P05177 1/20 0.50
CYP3A4 P08684 1/20 0.50
CYP2D6 P10635 1/20 0.50
CYP2C9 P11712 1/20 0.50
HTR2A P28223 1/20 0.50
SLC6A4 P31645 1/20 0.50
CYP2C19 P33261 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30087959 0.90 CHRNB2 (0.47) HTR7ADRB1HTR1AHTR3EHTR3B
SCHEMBL689422 0.89 HTR7 (0.62) HTR7ADRB1HTR1AHTR3EHTR3B
Hydrochloric Acid SCHEMBL4661519 0.87 HTR7 (0.61) HTR7ADRB1HTR1AHTR3EHTR3B
SCHEMBL5540575 0.79 ADRB1 (0.80) HTR7ADRB1HTR1AHTR3EHTR3B
SCHEMBL56706 0.77 ADRB1 (0.75) HTR7ADRB1HTR1AHTR3EHTR3B
SCHEMBL1353556 0.75 MEN1 (0.52) HTTALDH1A1MAPTMEN1KMT2A
SCHEMBL1699410 0.75 DHFR (0.50) ALDH1A1MEN1KMT2AALOX5
Ammonia Solution, Strong SCHEMBL20512352 0.75 ADRB1 (0.72) HTR7ADRB1HTR1AHTR3EHTR3B
Hydrochloric Acid SCHEMBL11019815 0.75 ADRB1 (0.72) HTR7ADRB1HTR1AHTR3EHTR3B
Water SCHEMBL28163332 0.75 ADRB1 (0.72) HTR7ADRB1HTR1AHTR3EHTR3B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105658640-A Alkynyl alcohols and methods of use 豪夫迈·罗氏有限公司 2016-06-08 CN disclosed