SCHEMBL28085547

SCHEMBL28085547

COc1ccc(-c2c(Nc3cc(OC)c(OC)c(OC)c3)c3ccc(OCc4ccccc4)cc3oc2=O)cc1

nearest known ligand 0.58

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.58
ALDH1A1 P00352 1/20 0.58
HPGD P15428 1/20 0.58
SMN1; SMN2 Q16637 1/20 0.58
MAOB P27338 8/20 0.51
ACHE P22303 2/20 0.51
ESR1 P03372 4/20 0.50
CYP19A1 P11511 3/20 0.50
MAOA P21397 2/20 0.48
TDP1 Q9NUW8 2/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28085534 0.86 ESR1 (0.57) MAOBACHEESR1CYP19A1MAOA
SCHEMBL28085701 0.85 MAOB (0.56) KDM4EALDH1A1HPGDSMN1; SMN2MAOB
SCHEMBL28085538 0.83 ESR1 (0.54) KDM4EALDH1A1SMN1; SMN2MAOBACHE
SCHEMBL28085675 0.79 MAOB (0.65) KDM4EALDH1A1SMN1; SMN2MAOBACHE
SCHEMBL28085539 0.75 CYP19A1 (0.59) KDM4EALDH1A1HPGDSMN1; SMN2MAOB
SCHEMBL28085548 0.72 ESR1 (0.73) KDM4EALDH1A1SMN1; SMN2ESR1
SCHEMBL26779874 0.72 MAOB (0.79) KDM4EALDH1A1MAOBACHEMAOA
SCHEMBL30667382 0.72 ABCG2 (0.58) KDM4EALDH1A1HPGDSMN1; SMN2MAOB
SCHEMBL6823769 0.71 MAOB (0.53) KDM4EALDH1A1HPGDMAOBACHE
SCHEMBL28085659 0.71 ESR1 (0.58) KDM4EALDH1A1HPGDMAOBESR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105801544-A 3-aryl-4-arylamine-coumarin derivative and preparing method and medical application thereof 中国药科大学 2016-07-27 CN disclosed