SCHEMBL28086120

SCHEMBL28086120

CN1CCN(c2ccc(-n3cccc3-c3cccc(S(F)(F)(F)(F)F)c3)cc2)CC1

nearest known ligand 0.46

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
FYN P06241 3/20 0.40
ADRA2C P18825 2/20 0.38
ALDH1A1 P00352 2/20 0.38
KDM4E B2RXH2 1/20 0.38
GAA P10253 1/20 0.38
MAPT P10636 1/20 0.38
GFER P55789 1/20 0.38
KMT2A Q03164 1/20 0.38
PTK2B Q14289 1/20 0.38
ESR2 Q92731 1/20 0.38
MAP4K1 Q92918 1/20 0.38
MELK Q14680 1/20 0.38
HTR3A P46098 1/20 0.38
JAK2 O60674 5/20 0.37
ASIC3 Q9UHC3 1/20 0.36
JAK3 P52333 4/20 0.36
PTK2 Q05397 4/20 0.36
ACVR1 Q04771 1/20 0.35
AOC3 Q16853 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13735233 0.78 MAP4K1 (0.42) FYNADRA2CALDH1A1KDM4EGAA
SCHEMBL18656564 0.75 ADRA2C (0.61) ADRA2CALDH1A1KDM4EGAAMAPT
SCHEMBL18656562 0.71 MAPT (0.59) ADRA2CALDH1A1KDM4EGAAMAPT
SCHEMBL13734373 0.67 PTGS2 (0.43) FYNALDH1A1KDM4EMAPTKMT2A
SCHEMBL28086177 0.66 SIGMAR1 (0.50) ADRA2CALDH1A1KDM4EMAPT
SCHEMBL30108226 0.65 MELK (0.60) ADRA2CALDH1A1KDM4EGAAMAPT
SCHEMBL24061151 0.64 MAPKAPK2 (0.58) ADRA2CALDH1A1KDM4EGAAMAPT
SCHEMBL28845811 0.62 ADRA2C (0.70) FYNADRA2CALDH1A1KDM4EGAA
SCHEMBL18642123 0.62 HTR7 (0.57) ALDH1A1MAPTHTR3A
SCHEMBL18656551 0.62 ADRA2C (0.42) ADRA2CALDH1A1MAPTHTR3A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-103492389-B Pyrazolo [4,3-d] pyrimidine as inhibitors of kinases 原真股份有限公司 2016-09-14 CN disclosed