SCHEMBL28087492

SCHEMBL28087492

CCC(C(=O)OC)c1cc(F)c(F)cc1F

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
POLB P06746 1/20 0.36
ESR1 P03372 1/20 0.35
ESR2 Q92731 1/20 0.35
DPP4 P27487 2/20 0.35
TAS1R3 Q7RTX0 1/20 0.35
TAS1R1 Q7RTX1 1/20 0.35
AKR1C3 P42330 6/20 0.34
AKR1C2 P52895 6/20 0.34
CHRNA1 P02708 1/20 0.33
CHRNG P07510 1/20 0.33
CHRNB1 P11230 1/20 0.33
CHRNB2 P17787 1/20 0.33
SLC6A2 P23975 1/20 0.33
CHRNB4 P30926 1/20 0.33
CHRNA3 P32297 1/20 0.33
CHRNA4 P43681 1/20 0.33
SLC6A3 Q01959 1/20 0.33
CHRND Q07001 1/20 0.33
CA1 P00915 1/20 0.33
CA2 P00918 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL536349 0.80 AKR1C3 (0.44) AKR1C3AKR1C2AKR1C1PTGS1
SCHEMBL30231208 0.80 AKR1C3 (0.44) AKR1C3AKR1C2AKR1C1PTGS1
SCHEMBL28135500 0.79 AKR1C3 (0.34) AKR1C3AKR1C2CA1CA2LMNA
SCHEMBL5082189 0.77 CES2 (0.35) DPP4CHRNA1CHRNGCHRNB1CHRNB2
SCHEMBL5082185 0.77 CES2 (0.35) DPP4CHRNA1CHRNGCHRNB1CHRNB2
SCHEMBL7882734 0.75 KMT2A (0.33) DPP4CHRNA1CHRNGCHRNB1CHRNB2
SCHEMBL5084418 0.75 PSEN1 (0.35) DPP4CHRNA1CHRNGCHRNB1CHRNB2
SCHEMBL28784595 0.74 MAPT (0.35) AKR1C3AKR1C2HPGDLMNAMAPT
SCHEMBL28435707 0.74 ALDH1A1 (0.35) DPP4CHRNA1CHRNGCHRNB1CHRNB2
SCHEMBL6904784 0.71 RORC (0.44) POLBCA1CA2HPGDLMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-102574856-B The synthesis of sitagliptin 基因里克斯(英国)有限公司 2016-09-21 CN disclosed