SCHEMBL28087665

SCHEMBL28087665

O=C(O)CCc1cn(C2CC2)c2c(OC(F)F)c(Br)ccc2c1=O

nearest known ligand 0.35

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 4/20 0.35
GSK3B P49841 2/20 0.33
PLA2G4A P47712 1/20 0.32
S1PR1 P21453 1/20 0.31
THRA P10827 1/20 0.31
THRB P10828 1/20 0.31
TOP2A P11388 2/20 0.30
TOP2B Q02880 2/20 0.30
SCD O00767 1/20 0.30
CHRM2 P08172 1/20 0.30
CHRM1 P11229 1/20 0.30
CHRM3 P20309 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2903740 0.82 KCNH2 (0.50) KCNH2GSK3BTOP2ATOP2B
SCHEMBL27898679 0.71 GSK3B (0.49) KCNH2GSK3BTOP2ATOP2B
SCHEMBL5734714 0.64 TOP2A (0.57) KCNH2GSK3BTOP2ATOP2B
SCHEMBL13927305 0.63 TOP2A (0.44) KCNH2GSK3BTOP2ATOP2B
SCHEMBL3720416 0.63 TOP2A (0.58) KCNH2GSK3BTOP2ATOP2BCHRM2
SCHEMBL27593515 0.61 KCNH2 (0.53) KCNH2GSK3BTOP2ATOP2BCHRM2
SCHEMBL4998742 0.61 KCNH2 (0.46) KCNH2GSK3BTOP2ATOP2B
SCHEMBL5142579 0.61 TOP2A (0.55) KCNH2GSK3BTOP2ATOP2BCHRM2
SCHEMBL28774485 0.61 MMP12 (0.35)
SCHEMBL7507103 0.60 ADRB2 (0.55) KCNH2TOP2ATOP2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105837555-A Preparation method for garenoxacin and intermediate thereof 南京华威医药科技开发有限公司 2016-08-10 CN disclosed