SCHEMBL28088002

SCHEMBL28088002

FC(F)(F)c1cnccn1.NNC=O

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 2/20 0.35
ALOX15 P16050 1/20 0.35
CASP1 P29466 1/20 0.35
NPSR1 Q6W5P4 1/20 0.35
HSD17B10 Q99714 1/20 0.35
HSP90AA1 P07900 1/20 0.33
CYP19A1 P11511 1/20 0.33
TRPV4 Q9HBA0 1/20 0.33
NPC1 O15118 1/20 0.33
RAB9A P51151 1/20 0.33
L3MBTL1 Q9Y468 1/20 0.33
KDM4E B2RXH2 3/20 0.33
LOXL2 Q9Y4K0 2/20 0.33
ADORA3 P0DMS8 1/20 0.32
MC4R P32245 1/20 0.32
ADRA1A P35348 1/20 0.32
MC3R P41968 1/20 0.32
LOX P28300 1/20 0.32
P4HB P07237 1/20 0.31
VNN1 O95497 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29526853 0.82 TRPV4 (0.44) TSHRALOX15CASP1NPSR1HSD17B10
SCHEMBL631338 0.82 TRPV4 (0.44) TSHRALOX15CASP1NPSR1HSD17B10
SCHEMBL28687790 0.81 CYP19A1 (0.33) TSHRALOX15CASP1NPSR1HSD17B10
SCHEMBL27976387 0.79 CA2 (0.36) TRPV4KDM4E
SCHEMBL28221312 0.79 RAB9A (0.34) TSHRALOX15CASP1NPSR1HSD17B10
SCHEMBL29193221 0.75 SMN1; SMN2 (0.42) L3MBTL1KDM4ELOXL2LOX
SCHEMBL27976684 0.74 TRPV4 (0.44) TRPV4
Ethoxycarbonyl Group SCHEMBL27906093 0.73 KMT2A (0.34) CYP19A1TRPV4NPC1RAB9AL3MBTL1
SCHEMBL27982440 0.73 HSP90AA1 (0.67) TSHRHSP90AA1NPC1RAB9AKDM4E
SCHEMBL27982915 0.72 ADORA3 (0.39) TSHRHSP90AA1NPC1RAB9AKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-103946221-B heterocyclic compounds for the treatment of cystic fibrosis 诺华股份有限公司 2016-08-03 CN disclosed