SCHEMBL28089401

SCHEMBL28089401

c1ccc(C2=NC(c3ccccc3)(c3ccc4ccccc4n3)N=C2c2ccccc2)cc1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTT P42858 2/20 0.37
NCF1 P14598 3/20 0.36
CYP1A2 P05177 2/20 0.36
NOS2 P35228 1/20 0.36
BACE1 P56817 1/20 0.36
CA12 O43570 1/20 0.36
CA9 Q16790 1/20 0.36
MGAM O43451 1/20 0.36
CYSLTR2 Q9NS75 1/20 0.36
CYSLTR1 Q9Y271 1/20 0.36
NPC1 O15118 4/20 0.35
RAB9A P51151 4/20 0.35
AR P10275 2/20 0.35
CYP3A4 P08684 2/20 0.35
CYP2D6 P10635 1/20 0.35
CYP2C9 P11712 1/20 0.35
CYP2C19 P33261 1/20 0.35
LMNA P02545 2/20 0.35
PKM P14618 3/20 0.34
MEN1 O00255 3/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL28015992 0.98 HTT (0.36) HTTNCF1CYP1A2NOS2BACE1
SCHEMBL491053 0.65 ALDH1A1 (0.39) HTTBACE1NPC1RAB9ACYP2C9
2-Phenylquinoline SCHEMBL44999 0.64 RAB9A (0.73) CYP1A2NPC1RAB9AARCYP3A4
2-Phenylquinoline SCHEMBL29399739 0.64 RAB9A (0.73) CYP1A2NPC1RAB9AARCYP3A4
SCHEMBL8666648 0.63 CYP1A1 (0.39) CYP1A2MEN1KMT2AKDM4EALDH1A1
2-Phenylquinoline SCHEMBL346742 0.62 RAB9A (0.70) CYP1A2NPC1RAB9AARCYP3A4
2-Phenylquinoline SCHEMBL6858671 0.62 RAB9A (0.70) CYP1A2NPC1RAB9AARCYP3A4
2-Phenylquinoline SCHEMBL1815021 0.62 RAB9A (0.70) CYP1A2NPC1RAB9AARCYP3A4
2-Phenylquinoline SCHEMBL5733254 0.62 RAB9A (0.70) CYP1A2NPC1RAB9AARCYP3A4
2-Phenylquinoline SCHEMBL28871326 0.62 RAB9A (0.70) CYP1A2NPC1RAB9AARCYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-103923067-B The micromolecular inhibitor of a kind of MdmX/Mdm2 and preparation method and application 湖北工业大学 2016-08-24 CN disclosed