SCHEMBL28089634

SCHEMBL28089634

O=C(O)c1cc(CCc2ccc(Br)cc2)cc(C(=O)O)c1

nearest known ligand 0.49

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
RXRA P19793 1/20 0.49
RXRB P28702 1/20 0.49
MRGPRX4 Q96LA9 1/20 0.47
POLB P06746 2/20 0.46
MEN1 O00255 1/20 0.46
KMT2A Q03164 1/20 0.46
COPS5 Q92905 1/20 0.45
GPR52 Q9Y2T5 1/20 0.45
PDPK1 O15530 1/20 0.45
CTDSP1 Q9GZU7 1/20 0.45
GAA P10253 1/20 0.42
FFAR1 O14842 1/20 0.42
FFAR4 Q5NUL3 1/20 0.42
HTR2A P28223 1/20 0.42
TAAR1 Q96RJ0 1/20 0.42
HDAC1 Q13547 1/20 0.42
DAO P14920 1/20 0.41
TTR P02766 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16749638 0.83 CA12 (0.48) MEN1KMT2AGAADAOTTR
SCHEMBL27766830 0.82 GAA (0.59) MEN1KMT2AGAAFFAR1HDAC1
SCHEMBL27633124 0.81 ALDH1A1 (0.64) RXRARXRBMEN1KMT2AGAA
SCHEMBL28069551 0.81 PTGS1 (0.50) FFAR1DAO
SCHEMBL28851716 0.80 MRGPRX4 (0.54) MRGPRX4FFAR1FFAR4TAAR1
SCHEMBL11684208 0.78 RXRA (0.46) RXRARXRBMRGPRX4POLBMEN1
SCHEMBL27646690 0.77 CA1 (0.58) MRGPRX4POLBFFAR1
SCHEMBL28170053 0.77 MRGPRX4 (0.49) MRGPRX4FFAR1HDAC1DAO
SCHEMBL11687234 0.76 RXRA (0.45) RXRARXRBMRGPRX4POLBMEN1
SCHEMBL14166175 0.76 DHODH (0.56) RXRARXRBMEN1KMT2AGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105777756-A Heteroaryl compound and application thereof in medicines 广东东阳光药业有限公司 2016-07-20 CN disclosed