SCHEMBL28093453

SCHEMBL28093453

CC1(C)OCC(Cc2cc3ccccc3s2)C(C(=O)C=O)O1

nearest known ligand 0.40

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CYP2A6 P11509 3/20 0.39
TBXA2R P21731 1/20 0.37
ADRB2 P07550 1/20 0.36
ASIC3 Q9UHC3 1/20 0.36
LOXL2 Q9Y4K0 1/20 0.36
DRD2 P14416 1/20 0.36
DRD4 P21917 1/20 0.36
DRD3 P35462 1/20 0.36
TBXAS1 P24557 1/20 0.36
FFAR2 O15552 1/20 0.36
BCL2L1 Q07817 1/20 0.35
SLC6A2 P23975 1/20 0.35
SLC6A4 P31645 1/20 0.35
SLC6A3 Q01959 1/20 0.35
ALOX5 P09917 1/20 0.34
AGXT P21549 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28061650 0.73 TMEM97 (0.35) TBXA2RTBXAS1
SCHEMBL28124735 0.73 HCRTR2 (0.38) TBXA2RTBXAS1
SCHEMBL28061679 0.72 P2RX3 (0.40)
SCHEMBL28125140 0.71 GLA (0.43)
SCHEMBL28061680 0.70 LTB4R (0.38) TBXA2RTBXAS1
SCHEMBL27809084 0.70 EGFR (0.39) TBXA2RTBXAS1
SCHEMBL27769694 0.70 HCRTR2 (0.44) TBXA2R
SCHEMBL28067355 0.68 MMP9 (0.44)
SCHEMBL28294382 0.67 TBXA2R (0.32) TBXA2RTBXAS1
SCHEMBL16460682 0.66 GLA (0.47) CYP2A6ADRB2ASIC3LOXL2BCL2L1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105829294-B The quinolyl conditioning agent of ROR- γ-T being connect with methylene 詹森药业有限公司 2018-11-09 CN disclosed
CN-105829294-A METHYLENE LINKED QUINOLINYL MODULATORS OF ROR-GAMMA-T 詹森药业有限公司 2016-08-03 CN disclosed