SCHEMBL28097299

SCHEMBL28097299

COC(=O)c1cccc(N2CC=Cc3ccccc32)c1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.49
LMNA P02545 1/20 0.49
MAPK1 P28482 1/20 0.49
GAA P10253 1/20 0.48
TP53 P04637 1/20 0.45
NPC1 O15118 1/20 0.44
HPGD P15428 3/20 0.44
RAB9A P51151 2/20 0.44
PMM2 O15305 1/20 0.44
MPI P34949 1/20 0.44
PHOSPHO1 Q8TCT1 1/20 0.44
OPRM1 P35372 1/20 0.43
OPRL1 P41146 1/20 0.43
CTSG P08311 1/20 0.42
CMA1 P23946 1/20 0.42
GRM2 Q14416 1/20 0.42
CYP1A2 P05177 1/20 0.42
CYP2D6 P10635 1/20 0.42
MAPT P10636 1/20 0.42
CYP2C19 P33261 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28016744 0.75 MTNR1A (0.40) ALDH1A1LMNAMAPK1MAPTTSHR
SCHEMBL28185358 0.74 MTNR1A (0.40) ALDH1A1LMNAMAPK1MAPTTSHR
SCHEMBL28158396 0.73 KCNH2 (0.41) OPRL1
SCHEMBL21815682 0.73 SIGMAR1 (0.38) ALDH1A1LMNAMAPK1GAATP53
SCHEMBL5801010 0.73 ALDH1A1 (0.42) ALDH1A1MAPK1TP53CYP1A2CYP2D6
SCHEMBL28158980 0.73 FAAH (0.40) ALDH1A1LMNAGAAOPRM1OPRL1
SCHEMBL32688194 0.72 ALDH1A1 (0.55) ALDH1A1LMNAMAPK1GAANPC1
SCHEMBL22028459 0.71 SIGMAR1 (0.36) ALDH1A1LMNAMAPK1GAATP53
SCHEMBL1408252 0.71 SIGMAR1 (0.36) ALDH1A1LMNAMAPK1GAATP53
SCHEMBL30919258 0.71 SIGMAR1 (0.36) ALDH1A1LMNAMAPK1GAATP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-104230827-B 1-(aryl methyl) quinazoline-2,4 (1H, 3H)-diketone is as PARP inhibitor and application thereof 南京英派药业有限公司 2016-10-26 CN disclosed