SCHEMBL28097813

SCHEMBL28097813

COOB(O)c1ccncc1

nearest known ligand 0.32

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 2/20 0.32
CYP2C9 P11712 2/20 0.32
CYP2C19 P33261 2/20 0.32
SMN1; SMN2 Q16637 2/20 0.32
LMNA P02545 2/20 0.32
KDM4E B2RXH2 1/20 0.31
NPC1 O15118 1/20 0.31
CYP3A4 P08684 1/20 0.31
CYP2D6 P10635 1/20 0.31
HPGD P15428 1/20 0.31
RAB9A P51151 1/20 0.31
CA1 P00915 1/20 0.31
CA2 P00918 1/20 0.31
ENPP2 Q13822 1/20 0.31
MAPT P10636 1/20 0.31
KIF11 P52732 1/20 0.30
ERN1 O75460 1/20 0.30
CHRM5 P08912 1/20 0.30
CHKA P35790 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16825623 0.82 CYP1A2 (0.33) CYP1A2CYP2C9CYP2C19SMN1; SMN2LMNA
SCHEMBL262207 0.77 ENPP2 (0.46) CA1CA2ENPP2
SCHEMBL4716676 0.76 HSP90AA1 (0.33)
SCHEMBL568870 0.76 ALDH1A1 (0.41) CYP1A2CYP2C19SMN1; SMN2LMNAKDM4E
Fluoride SCHEMBL28835775 0.76 ENPP2 (0.44) CA1CA2ENPP2
SCHEMBL14066349 0.75 LMNA (0.35) CYP1A2CYP2C9CYP2C19SMN1; SMN2LMNA
SCHEMBL16429084 0.74 ERN1 (0.30) ERN1
SCHEMBL26924069 0.74 ORAI1 (0.50) KDM4ENPC1RAB9ACA1CA2
SCHEMBL26924303 0.74 TRPV6 (0.55) CA1CA2KIF11
SCHEMBL1485477 0.73 USP2 (0.34) CYP1A2CYP2C9CYP2C19SMN1; SMN2LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-104755478-B Serine/threonine kinase inhibitor 霍夫曼-拉罗奇有限公司 2017-10-10 CN disclosed
CN-103384672-B The substituted piperazine of N-pteridine and piperazine pteridinone 武田药品工业株式会社 2016-09-28 CN disclosed