SCHEMBL28100693

SCHEMBL28100693

O=COc1c(F)cccc1Br

nearest known ligand 0.36

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
EPAS1 Q99814 1/20 0.36
ERN1 O75460 1/20 0.34
MAOB P27338 1/20 0.33
HTT P42858 1/20 0.33
GCK P35557 1/20 0.31
CES2 O00748 1/20 0.31
CES1 P23141 1/20 0.31
KRAS P01116 1/20 0.30
CYP2A6 P11509 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1992255 0.85 ERN1 (0.40) ERN1CES2CES1KRAS
SCHEMBL16545836 0.76 KMT2A (0.40) ERN1
SCHEMBL589662 0.72 KRAS (0.39) EPAS1HTTGCKKRAS
SCHEMBL10209572 0.72 ALDH1A1 (0.30) CYP2A6
SCHEMBL28873828 0.72 DYRK1A (0.38) HTT
SCHEMBL6442207 0.72 ALB (0.52) CES2CES1
SCHEMBL24207668 0.72 RAB9A (0.34) ERN1HTTGCK
SCHEMBL21369287 0.72 HPGD (0.35) HTT
SCHEMBL25181496 0.71 CA1 (0.37)
SCHEMBL1997466 0.70 CES2 (0.38) ERN1CES2CES1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-103958504-B 10A type phosphodiesterase inhibitor compound 艾伯维德国有限责任两合公司 2016-10-12 CN disclosed