SCHEMBL28102575

SCHEMBL28102575

NC(=O)N1CC(=O)Nc2cc(C(=O)O)ccc21

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTT P42858 3/20 0.49
BRD4 O60885 6/20 0.47
BRD2 P25440 3/20 0.47
TUBB4A P04350 1/20 0.47
TUBB P07437 1/20 0.47
TUBA3C P0DPH7 1/20 0.47
TUBA1B P68363 1/20 0.47
TUBA4A P68366 1/20 0.47
TUBB4B P68371 1/20 0.47
TUBB3 Q13509 1/20 0.47
TUBB2A Q13885 1/20 0.47
TUBB8 Q3ZCM7 1/20 0.47
TUBA3E Q6PEY2 1/20 0.47
TUBA1A Q71U36 1/20 0.47
TUBA1C Q9BQE3 1/20 0.47
TUBB6 Q9BUF5 1/20 0.47
TUBB2B Q9BVA1 1/20 0.47
TUBB1 Q9H4B7 1/20 0.47
MEN1 O00255 2/20 0.47
KMT2A Q03164 2/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL26348154 0.81 ALDH1A1 (0.46) HTTBRD4BRD2TUBB4ATUBB
SCHEMBL30860393 0.79 HTT (0.49) HTTBRD4BRD2TUBB4ATUBB
SCHEMBL3803421 0.79 HTT (0.49) HTTBRD4BRD2TUBB4ATUBB
SCHEMBL18660612 0.71 HTT (0.80) HTTBRD4BRD2MEN1KMT2A
SCHEMBL31518440 0.68 HTT (0.57) HTTPOLBSMN1; SMN2L3MBTL1GAA
SCHEMBL21606267 0.68 NR1H2 (0.43) HTTMEN1KMT2AALDH1A1LMNA
SCHEMBL31539452 0.68 MAPK1 (0.49) HTTBRD4BRD2TUBB4ATUBB
SCHEMBL398818 0.67 TDP2 (0.66) HTTALDH1A1GAA
SCHEMBL29713338 0.67 TDP2 (0.66) HTTALDH1A1GAA
SCHEMBL26338105 0.67 AMPD2 (0.40) HTTBRD4ALDH1A1PARP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-106146416-B Nitrogen replaces 3- oxo -6- substituted-tetrahydro quinoxaline structural compounds, preparation method and its medical usage 河南大学 2019-02-19 CN disclosed
CN-106146416-A Nitrogen replaces 3 oxo 6 substituted-tetrahydro quinoxaline structural compounds, its preparation method and medical usage thereof 河南大学 2016-11-23 CN disclosed