SCHEMBL28109727

SCHEMBL28109727

FC(F)(F)c1cccc(N2CCc3cccnc32)c1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.56
MAPT P10636 3/20 0.56
KDM4E B2RXH2 3/20 0.56
ALOX5 P09917 2/20 0.49
PTGS1 P23219 1/20 0.49
PTGS2 P35354 1/20 0.49
HTR3E A5X5Y0 1/20 0.43
HTR3B O95264 1/20 0.43
HTR1D P28221 1/20 0.43
HTR2C P28335 1/20 0.43
HTR3A P46098 1/20 0.43
HTR3D Q70Z44 1/20 0.43
HTR3C Q8WXA8 1/20 0.43
SIGMAR1 Q99720 1/20 0.43
DRD2 P14416 1/20 0.43
DRD3 P35462 1/20 0.43
KCNH2 Q12809 1/20 0.43
LMNA P02545 1/20 0.43
HTT P42858 1/20 0.43
NPSR1 Q6W5P4 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30900480 0.74 NUDT1 (0.39) PHGDHNUDT1
SCHEMBL11733576 0.73 MEN1 (0.48) ALDH1A1MAPTKDM4EALOX5HTR3E
SCHEMBL432973 0.72 ALOX5 (0.55) ALDH1A1MAPTKDM4EALOX5PTGS1
SCHEMBL2479231 0.71 ALDH1A1 (0.51) ALDH1A1MAPTKDM4EALOX5PTGS1
SCHEMBL11728248 0.70 DRD3 (0.43) ALDH1A1MAPTKDM4EDRD2DRD3
SCHEMBL11729992 0.70 PIK3CA (0.50) ALDH1A1DRD2DRD3KCNH2HTT
SCHEMBL10539432 0.69 ALDH1A1 (0.79) ALDH1A1MAPTKDM4EALOX5PTGS1
SCHEMBL18003260 0.68 ALDH1A1 (0.51) ALDH1A1MAPTKDM4EALOX5PTGS1
SCHEMBL11732890 0.68 DRD2 (0.43) ALDH1A1DRD2DRD3KCNH2HTT
SCHEMBL15766789 0.68 DDB1 (0.64) ALDH1A1MAPTKDM4EALOX5PTGS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-102725291-B Bicyclic pyridine and relevant analog as Sirtuin regulator 西特里斯药业公司 2016-12-21 CN disclosed