SCHEMBL28111917

SCHEMBL28111917

c1ccc(-c2nccn2On2ccnc2-c2ccccc2)cc1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 1/20 0.45
CHEK1 O14757 2/20 0.40
ALDH1A1 P00352 2/20 0.40
LIMK1 P53667 2/20 0.40
MAPK14 Q16539 2/20 0.40
KDM4E B2RXH2 1/20 0.40
MAPT P10636 1/20 0.40
TDP1 Q9NUW8 1/20 0.40
KDR P35968 10/20 0.40
PRKACA P17612 2/20 0.39
CDK8 P49336 2/20 0.39
MAP2K1 Q02750 2/20 0.39
ACVR1 Q04771 2/20 0.39
ROCK1 Q13464 2/20 0.39
DYRK1B Q9Y463 2/20 0.39
MAP4K4 O95819 1/20 0.39
CSF1R P07333 1/20 0.39
MAP4K2 Q12851 1/20 0.39
DYRK1A Q13627 1/20 0.39
AURKB Q96GD4 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27495941 0.77 ESR1 (0.44) ESR1KDRPLAAALPG
SCHEMBL28062022 0.76 PARL (0.42) ESR1ALDH1A1KDM4EMAPTTDP1
SCHEMBL5192672 0.76 ESR1 (0.49) ESR1CHEK1ALDH1A1LIMK1MAPK14
SCHEMBL19065614 0.72 ESR1 (0.46) ESR1CHEK1ALDH1A1LIMK1MAPK14
SCHEMBL1263722 0.72 ESR1 (0.50) ESR1CHEK1ALDH1A1LIMK1MAPK14
SCHEMBL4482636 0.72 ESR1 (0.46) ESR1CHEK1ALDH1A1LIMK1MAPK14
SCHEMBL5533567 0.72 ESR1 (0.46) ESR1CHEK1ALDH1A1LIMK1MAPK14
SCHEMBL786747 0.72 HDAC4 (0.52) ESR1CHEK1ALDH1A1LIMK1MAPK14
SCHEMBL5324352 0.72 ESR1 (0.46) ESR1CHEK1ALDH1A1LIMK1MAPK14
SCHEMBL6440778 0.72 KMT2A (0.50) ESR1CHEK1ALDH1A1LIMK1MAPK14

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-106471032-A Catalyst for synthesizing oxazolidinone compound 科思创德国股份有限公司 2017-03-01 CN disclosed