SCHEMBL28113663

SCHEMBL28113663

O=COC(Cc1cc(O)[nH]n1)Cc1cccc(F)c1F

nearest known ligand 0.38

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
AKR1B1 P15121 2/20 0.38
PRKACA P17612 2/20 0.32
PRKACG P22612 2/20 0.32
PRKACB P22694 2/20 0.32
AKT1 P31749 2/20 0.32
ADORA2A P29274 1/20 0.32
ADORA1 P30542 1/20 0.32
DPP4 P27487 1/20 0.32
PIN1 Q13526 1/20 0.31
CXCR2 P25025 3/20 0.31
DYRK1A Q13627 1/20 0.31
CCR7 P32248 1/20 0.31
MPO P05164 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28325986 0.91 HCAR3 (0.34) AKR1B1DPP4
SCHEMBL28113597 0.84 AKR1B1 (0.36) AKR1B1PRKACAPRKACGPRKACBAKT1
SCHEMBL28113598 0.78 CTSK (0.34)
SCHEMBL27485646 0.77 DPP4 (0.34) AKR1B1AKT1DPP4MPO
SCHEMBL27627222 0.75 HCAR3 (0.30)
SCHEMBL28325982 0.74 HCAR3 (0.34) AKR1B1DPP4
SCHEMBL28327134 0.74 AKR1B1 (0.32) AKR1B1DPP4
SCHEMBL28113601 0.74 XPO1 (0.35)
SCHEMBL28113602 0.73
SCHEMBL27977725 0.71 AKR1B1 (0.33) AKR1B1DPP4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-106304835-A Sgc stimulant 铁木医药有限公司 2017-01-04 CN disclosed