SCHEMBL28114028

SCHEMBL28114028

CCC(=O)c1cc(Cl)c(Cl)c(I)c1OC

nearest known ligand 0.41

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
HMGCR P04035 1/20 0.41
L3MBTL1 Q9Y468 1/20 0.40
ALDH1A1 P00352 3/20 0.37
KDM4E B2RXH2 3/20 0.37
GAA P10253 1/20 0.37
HPGD P15428 1/20 0.35
PPARG P37231 1/20 0.34
PPARA Q07869 1/20 0.34
TPMT P51580 1/20 0.34
HSP90AA1 P07900 2/20 0.34
HSD17B10 Q99714 1/20 0.33
HSP90AB1 P08238 1/20 0.33
POLB P06746 1/20 0.33
DRD2 P14416 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9928852 0.82 ABCB11 (0.37) ALDH1A1KDM4EGAAHPGDTPMT
SCHEMBL9928867 0.74 L3MBTL1 (0.45) HMGCRL3MBTL1ALDH1A1KDM4EGAA
SCHEMBL1262272 0.72 PDE4D (0.43) HMGCRL3MBTL1ALDH1A1KDM4EGAA
SCHEMBL28114021 0.72 LMNA (0.38) HMGCRALDH1A1KDM4EGAAHPGD
SCHEMBL10994734 0.71 KDM4E (0.54) HMGCRL3MBTL1ALDH1A1KDM4EHPGD
SCHEMBL9720581 0.71 ALDH1A1 (0.49) HMGCRL3MBTL1ALDH1A1KDM4EGAA
SCHEMBL8895935 0.70 HMGCR (0.54) HMGCRALDH1A1GAA
SCHEMBL10994738 0.70 KDM4E (0.44) HMGCRL3MBTL1ALDH1A1KDM4EGAA
SCHEMBL28113489 0.70 LMNA (0.39) HMGCRL3MBTL1ALDH1A1KDM4EGAA
SCHEMBL12813097 0.69 CYP1A2 (0.35) ALDH1A1KDM4EGAATPMT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-104024253-B Heterocyclic amines as PI3K inhibitors INCYTE HOLDINGS CORP. (US) 2016-11-30 CN disclosed