SCHEMBL28115620

SCHEMBL28115620

C1=NN(c2cccnc2)CN1c1ccccc1

nearest known ligand 0.42

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
HTT P42858 2/20 0.41
MAPT P10636 1/20 0.41
MAPK1 P28482 1/20 0.41
CYP2A6 P11509 2/20 0.40
CYP3A4 P08684 1/20 0.40
CHRNB2 P17787 5/20 0.39
CHRNA4 P43681 5/20 0.39
CFTR P13569 1/20 0.39
SLC6A2 P23975 1/20 0.39
SLC6A4 P31645 1/20 0.39
SLC6A3 Q01959 1/20 0.39
GOPC Q9HD26 1/20 0.39
CHRNB4 P30926 1/20 0.39
CHRNA3 P32297 1/20 0.39
CYP11B2 P19099 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3861449 0.85 MAPT (0.41) HTTMAPTMAPK1CYP3A4
SCHEMBL28115615 0.76 MAOB (0.47) HTTMAPTMAPK1CYP3A4
SCHEMBL28115962 0.73 KEAP1 (0.38) MAPT
SCHEMBL30720445 0.71 CHRNB2 (0.45) HTTMAPTMAPK1CYP2A6CYP3A4
SCHEMBL27557204 0.71 CHRNB2 (0.42) HTTMAPTMAPK1CYP2A6CYP3A4
SCHEMBL2731119 0.69 MAPT (0.73) HTTMAPTMAPK1CHRNB2CHRNA4
SCHEMBL21864339 0.68 SMN1; SMN2 (0.38) MAPTMAPK1CYP3A4CHRNB2CHRNA4
SCHEMBL28252032 0.67 LMNA (0.37) HTTCHRNA4SLC6A2SLC6A4SLC6A3
Iodide SCHEMBL27085276 0.67 NPC1 (0.37) MAPTMAPK1CYP3A4CHRNB2CHRNA4
SCHEMBL29366505 0.67 CYP2A6 (0.44) HTTMAPTCYP2A6CYP3A4CHRNB2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-106234385-B A kind of application of 1,2,4- triazole derivatives of the structure containing benzopyrazines as fungicide 浙江工业大学 2018-11-13 CN disclosed
CN-106432245-B A kind of 1,2,4- triazole derivatives of the structure containing benzopyrazines and its preparation method and application 浙江工业大学 2018-11-13 CN disclosed
CN-106432245-A 1,2,4-triazole derivative having quinoxaline structure, preparation method and application thereof 浙江工业大学 2017-02-22 CN disclosed
CN-106234385-A A kind of 1,2,4 triazole derivatives containing benzopyrazines structure are as the application of antibacterial 浙江工业大学 2016-12-21 CN disclosed