SCHEMBL28115969

SCHEMBL28115969

NCCS(=O)(=O)NC(=O)c1cccnc1

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 5/20 0.57
HDAC1 Q13547 2/20 0.57
HDAC6 Q9UBN7 1/20 0.57
THRB P10828 1/20 0.56
PTGS1 P23219 2/20 0.53
EGFR P00533 2/20 0.53
HDAC3 O15379 1/20 0.50
HDAC2 Q92769 1/20 0.50
LMNA P02545 1/20 0.49
HIF1A Q16665 1/20 0.49
CYP3A4 P08684 3/20 0.48
ROCK2 O75116 1/20 0.48
ROCK1 Q13464 1/20 0.48
F7 P08709 1/20 0.47
F3 P13726 1/20 0.47
SARM1 Q6SZW1 1/20 0.47
SIRT2 Q8IXJ6 1/20 0.47
SIRT6 Q8N6T7 1/20 0.47
SIRT1 Q96EB6 1/20 0.47
SIRT3 Q9NTG7 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28116378 0.92 PTGS2 (0.55) PTGS2HDAC1HDAC6THRBPTGS1
SCHEMBL30437125 0.85 PTGS2 (0.57) PTGS2HDAC1HDAC6THRBPTGS1
SCHEMBL28115972 0.81 PTGS2 (0.52) PTGS2HDAC1HDAC6THRBPTGS1
SCHEMBL6131014 0.78 HDAC1 (0.54) HDAC1HDAC6HDAC3HDAC2LMNA
SCHEMBL1820805 0.76 HDAC1 (0.66) PTGS2HDAC1HDAC6THRBPTGS1
SCHEMBL11864560 0.76 HDAC1 (0.66) PTGS2HDAC1HDAC6THRBPTGS1
Nicotinic Acid Hydrazide SCHEMBL258390 0.76 HDAC1 (0.69) HDAC1HDAC6THRBHDAC3HDAC2
Nicotinic Acid Hydrazide SCHEMBL29648965 0.76 HDAC1 (0.69) HDAC1HDAC6THRBHDAC3HDAC2
SCHEMBL732195 0.75 THRB (0.68) HDAC1HDAC6THRBCYP3A4CYP2C9
SCHEMBL15625506 0.75 KMT2A (0.59) THRBCYP3A4CYP2C9MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-104478798-B N-aminoalkyl-3-pyridinecarboxamide derivative and application of N-aminoalkyl-3-pyridinecarboxamide derivative in preparation of drugs for treating cardiovascular and cerebrovascular diseases 武汉华纳联合药业有限公司 2017-01-18 CN claimed
CN-104478798-B N-aminoalkyl-3-pyridinecarboxamide derivative and application of N-aminoalkyl-3-pyridinecarboxamide derivative in preparation of drugs for treating cardiovascular and cerebrovascular diseases 武汉华纳联合药业有限公司 2017-01-18 CN disclosed