SCHEMBL28115972

SCHEMBL28115972

NCC(N)CS(=O)(=O)NC(=O)c1cccnc1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 5/20 0.52
HDAC1 Q13547 2/20 0.51
HDAC6 Q9UBN7 1/20 0.51
THRB P10828 1/20 0.51
PTGS1 P23219 2/20 0.49
EGFR P00533 2/20 0.49
PLOD2 O00469 1/20 0.46
LMNA P02545 1/20 0.44
HIF1A Q16665 1/20 0.44
CYP3A4 P08684 3/20 0.44
MEN1 O00255 3/20 0.44
KMT2A Q03164 3/20 0.44
ROCK2 O75116 1/20 0.43
ROCK1 Q13464 1/20 0.43
CYP2C9 P11712 2/20 0.43
CYP1A2 P05177 1/20 0.43
CYP2C19 P33261 1/20 0.43
EPHX2 P34913 1/20 0.43
HDAC3 O15379 1/20 0.43
HDAC2 Q92769 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28115969 0.81 PTGS2 (0.57) PTGS2HDAC1HDAC6THRBPTGS1
SCHEMBL28116378 0.78 PTGS2 (0.55) PTGS2HDAC1HDAC6THRBPTGS1
SCHEMBL28816391 0.77 PTGS2 (0.45) PTGS2HDAC1HDAC6THRBPTGS1
SCHEMBL30437125 0.75 PTGS2 (0.57) PTGS2HDAC1HDAC6THRBPTGS1
SCHEMBL28116024 0.73 ALDH1A1 (0.46) PTGS2HDAC1HDAC6THRBPTGS1
SCHEMBL11864560 0.72 HDAC1 (0.66) PTGS2HDAC1HDAC6THRBPTGS1
SCHEMBL1820805 0.72 HDAC1 (0.66) PTGS2HDAC1HDAC6THRBPTGS1
Nicotinic Acid Hydrazide SCHEMBL258390 0.71 HDAC1 (0.69) HDAC1HDAC6THRBPLOD2LMNA
Nicotinic Acid Hydrazide SCHEMBL29648965 0.71 HDAC1 (0.69) HDAC1HDAC6THRBPLOD2LMNA
SCHEMBL10894691 0.71 LMNA (0.65) HDAC1HDAC6THRBLMNAHIF1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-104478798-B N-aminoalkyl-3-pyridinecarboxamide derivative and application of N-aminoalkyl-3-pyridinecarboxamide derivative in preparation of drugs for treating cardiovascular and cerebrovascular diseases 武汉华纳联合药业有限公司 2017-01-18 CN claimed
CN-104478798-B N-aminoalkyl-3-pyridinecarboxamide derivative and application of N-aminoalkyl-3-pyridinecarboxamide derivative in preparation of drugs for treating cardiovascular and cerebrovascular diseases 武汉华纳联合药业有限公司 2017-01-18 CN disclosed