SCHEMBL28116024

SCHEMBL28116024

CCC(CNC(C)C)CS(=O)(=O)NC(=O)c1cccnc1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.46
NPC1 O15118 3/20 0.46
RAB9A P51151 3/20 0.46
SMN1; SMN2 Q16637 3/20 0.46
TP53 P04637 2/20 0.46
NPSR1 Q6W5P4 1/20 0.46
PTGS2 P35354 5/20 0.46
EGFR P00533 2/20 0.46
GAA P10253 2/20 0.46
THRB P10828 1/20 0.45
MEN1 O00255 3/20 0.45
KMT2A Q03164 3/20 0.45
HDAC1 Q13547 2/20 0.45
HDAC6 Q9UBN7 1/20 0.45
PTGS1 P23219 2/20 0.44
HDAC3 O15379 1/20 0.42
HDAC2 Q92769 1/20 0.42
LMNA P02545 1/20 0.41
CYP1A2 P05177 1/20 0.41
CYP3A4 P08684 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27996515 0.80 ALDH1A1 (0.43) ALDH1A1NPC1RAB9ASMN1; SMN2TP53
SCHEMBL30437125 0.75 PTGS2 (0.57) ALDH1A1NPC1RAB9ASMN1; SMN2NPSR1
SCHEMBL28115972 0.73 PTGS2 (0.52) NPC1RAB9ASMN1; SMN2PTGS2EGFR
SCHEMBL9809554 0.70 HDAC1 (0.57) ALDH1A1NPC1RAB9ASMN1; SMN2TP53
SCHEMBL29995369 0.70 ECE1 (0.60) ALDH1A1NPC1RAB9ASMN1; SMN2TP53
SCHEMBL24267375 0.70 ECE1 (0.60) ALDH1A1NPC1RAB9ASMN1; SMN2TP53
SCHEMBL3854614 0.70 KMT2A (0.63) ALDH1A1NPC1RAB9ASMN1; SMN2TP53
SCHEMBL1820805 0.70 HDAC1 (0.66) ALDH1A1PTGS2EGFRTHRBMEN1
SCHEMBL28115969 0.70 PTGS2 (0.57) NPC1RAB9ASMN1; SMN2PTGS2EGFR
SCHEMBL5553293 0.70 KMT2A (0.66) ALDH1A1NPC1RAB9ASMN1; SMN2TP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-104478798-B N-aminoalkyl-3-pyridinecarboxamide derivative and application of N-aminoalkyl-3-pyridinecarboxamide derivative in preparation of drugs for treating cardiovascular and cerebrovascular diseases 武汉华纳联合药业有限公司 2017-01-18 CN claimed
CN-104478798-B N-aminoalkyl-3-pyridinecarboxamide derivative and application of N-aminoalkyl-3-pyridinecarboxamide derivative in preparation of drugs for treating cardiovascular and cerebrovascular diseases 武汉华纳联合药业有限公司 2017-01-18 CN disclosed