SCHEMBL28118828

SCHEMBL28118828

CC(C)CCC1(O)C(=O)Nc2ccc(Nc3cccc(C(F)(F)F)c3)cc21

nearest known ligand 0.48

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
KIF11 P52732 11/20 0.48
TP53 P04637 1/20 0.43
NQO2 P16083 1/20 0.43
SMN1; SMN2 Q16637 2/20 0.42
KDM4E B2RXH2 1/20 0.42
AKR1C3 P42330 1/20 0.41
AKR1C2 P52895 1/20 0.41
GSK3B P49841 1/20 0.40
DHODH Q02127 1/20 0.40
HTT P42858 1/20 0.39
YAP1 P46937 1/20 0.39
TEAD4 Q15561 1/20 0.39
TEAD2 Q15562 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28119235 0.85 KIF11 (0.48) KIF11TP53NQO2AKR1C3AKR1C2
SCHEMBL28118830 0.84 KIF11 (0.47) KIF11TP53NQO2AKR1C3AKR1C2
SCHEMBL28119199 0.82 KIF11 (0.50) KIF11AKR1C3AKR1C2HTTYAP1
SCHEMBL28118836 0.80 NQO2 (0.47) NQO2GSK3B
SCHEMBL28119198 0.67 NQO2 (0.47) NQO2GSK3BHTT
SCHEMBL1921482 0.66 KIF11 (0.70) KIF11TP53SMN1; SMN2AKR1C3AKR1C2
SCHEMBL394991 0.66 KIF11 (0.70) KIF11SMN1; SMN2KDM4EAKR1C3AKR1C2
SCHEMBL28119197 0.66 NQO2 (0.46) NQO2GSK3BHTT
SCHEMBL16208518 0.66 KIF11 (1.00) KIF11AKR1C3AKR1C2
SCHEMBL4937177 0.65 KIF11 (0.56) KIF11TP53SMN1; SMN2KDM4EDHODH

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-106316923-A Disubstituted indol-2(1H)-one derivative and preparation method and application thereof 中南大学 2017-01-11 CN claimed
CN-106316923-A Disubstituted indol-2(1H)-one derivative and preparation method and application thereof 中南大学 2017-01-11 CN disclosed