SCHEMBL28118830

SCHEMBL28118830

CCCCCCC1(O)C(=O)Nc2ccc(Nc3cccc(C(F)(F)F)c3)cc21

nearest known ligand 0.47

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
KIF11 P52732 12/20 0.47
NQO2 P16083 1/20 0.42
HTR7 P34969 1/20 0.41
AKR1C3 P42330 1/20 0.40
AKR1C2 P52895 1/20 0.40
RXFP1 Q9HBX9 1/20 0.40
SPHK2 Q9NRA0 1/20 0.39
SPHK1 Q9NYA1 1/20 0.39
HTT P42858 2/20 0.38
YAP1 P46937 1/20 0.38
TEAD4 Q15561 1/20 0.38
TEAD2 Q15562 1/20 0.38
MEN1 O00255 1/20 0.38
LMNA P02545 1/20 0.38
TP53 P04637 1/20 0.38
MAPT P10636 1/20 0.38
ALOX15 P16050 1/20 0.38
MAPK1 P28482 1/20 0.38
KMT2A Q03164 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28119235 0.99 KIF11 (0.48) KIF11NQO2HTR7AKR1C3AKR1C2
SCHEMBL28118828 0.84 KIF11 (0.48) KIF11NQO2AKR1C3AKR1C2HTT
SCHEMBL28119197 0.83 NQO2 (0.46) NQO2HTR7HTTMEN1MAPT
SCHEMBL28119198 0.82 NQO2 (0.47) NQO2HTR7HTTMEN1MAPT
SCHEMBL28119199 0.81 KIF11 (0.50) KIF11AKR1C3AKR1C2RXFP1HTT
SCHEMBL28118909 0.81 NQO2 (0.46) NQO2HTR7HTTMEN1LMNA
SCHEMBL250063 0.69 GAA (0.54) HTTMEN1LMNAMAPTKMT2A
SCHEMBL25590656 0.67 LMNA (0.54) RXFP1SPHK2SPHK1MEN1LMNA
SCHEMBL17817420 0.66 HDAC3 (0.78) RXFP1MEN1LMNATP53MAPT
SCHEMBL31129776 0.66 HDAC3 (0.78) RXFP1MEN1LMNATP53MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-106316923-A Disubstituted indol-2(1H)-one derivative and preparation method and application thereof 中南大学 2017-01-11 CN claimed
CN-106316923-A Disubstituted indol-2(1H)-one derivative and preparation method and application thereof 中南大学 2017-01-11 CN disclosed