SCHEMBL28129013

SCHEMBL28129013

c1ccc(COc2ccccc2-c2cc[nH]n2)cc1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BRD4 O60885 4/20 0.54
IDO1 P14902 1/20 0.52
PDE5A O76074 1/20 0.47
PDE4A P27815 1/20 0.47
PDE4B Q07343 1/20 0.47
PDE4C Q08493 1/20 0.47
PDE4D Q08499 1/20 0.47
CNR1 P21554 1/20 0.46
CNR2 P34972 1/20 0.46
MAPT P10636 1/20 0.46
MAPK1 P28482 1/20 0.46
TDP1 Q9NUW8 1/20 0.46
L3MBTL1 Q9Y468 1/20 0.46
LTA4H P09960 1/20 0.45
MAPK14 Q16539 1/20 0.45
SGMS2 Q8NHU3 1/20 0.44
HTR1A P08908 1/20 0.44
DRD2 P14416 1/20 0.44
TLR4 O00206 1/20 0.43
TLR3 O15455 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28866549 0.84 MAOB (0.49) MAPTMAPK1TDP1L3MBTL1TLR9
SCHEMBL6028879 0.83 PTGER1 (0.53) PTGER1
SCHEMBL6452344 0.81 TLR9 (0.51) MAPTMAPK1HTR1ADRD2TLR9
SCHEMBL6448897 0.81 MAOB (0.48) BRD4HTR1ADRD2TLR9TLR7
SCHEMBL11625444 0.80 ALDH1A1 (0.50) PDE5AMAPTTDP1L3MBTL1
SCHEMBL3103763 0.80 L3MBTL1 (0.44) BRD4IDO1L3MBTL1PTGER1
SCHEMBL15825571 0.79 POLB (0.51) TDP1L3MBTL1
SCHEMBL26013299 0.78 MAPT (0.63) BRD4IDO1MAPTMAPK1TDP1
SCHEMBL14863659 0.77 LMNA (0.37) IDO1PDE5APDE4APDE4BPDE4C
SCHEMBL28284772 0.77 ADRA1D (0.58) BRD4IDO1PDE5APDE4APDE4B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-103476252-B Pyrazolyl guanidine F1F 0-ATPase inhibitors and therapeutic uses thereof 莱斯拉公司 2017-02-22 CN disclosed