SCHEMBL28146547

SCHEMBL28146547

COS(=O)(=O)O.Cc1cccc2nc3ccccc3cc12

nearest known ligand 0.45

Known targets — ChEMBL curated mechanism

ACHECHRM1CHRM3

The experimentally established mechanism targets of None. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ACHE known ✓ P22303 1/20 0.40
ALDH1A1 P00352 5/20 0.45
KDM4E B2RXH2 4/20 0.45
HPGD P15428 3/20 0.45
GLA P06280 2/20 0.45
GAA P10253 2/20 0.45
POLB P06746 2/20 0.45
KMT2A Q03164 2/20 0.45
NPC1 O15118 1/20 0.45
LMNA P02545 1/20 0.45
PTBP1 P26599 1/20 0.45
RAB9A P51151 1/20 0.45
RCE1 Q9Y256 1/20 0.45
PDE10A Q9Y233 1/20 0.41
PDE3B Q13370 2/20 0.40
PDE3A Q14432 2/20 0.40
MAPT P10636 1/20 0.40
RXFP1 Q9HBX9 1/20 0.39
TDP1 Q9NUW8 1/20 0.39
STAT3 P40763 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL38662128 0.85 TSHR (0.47) ALDH1A1KDM4EHPGDGLAGAA
Acridine SCHEMBL2823221 0.84 ALDH1A1 (0.58) ALDH1A1KDM4EHPGDGLAGAA
Trifluoromethanesulfonic Acid SCHEMBL3855068 0.84 ALDH1A1 (0.44) ALDH1A1KDM4EHPGDGLAGAA
SCHEMBL29376451 0.84 ALDH1A1 (0.60) ALDH1A1KDM4EHPGDGLAGAA
SCHEMBL291182 0.84 ALDH1A1 (0.60) ALDH1A1KDM4EHPGDGLAGAA
Hydrochloric Acid SCHEMBL28881738 0.82 ALDH1A1 (0.58) ALDH1A1KDM4EHPGDGLAGAA
SCHEMBL5854489 0.81 ALDH1A1 (0.53) ALDH1A1KDM4EHPGDGLAGAA
Nitric Acid SCHEMBL27968557 0.79 KMT2A (0.49) ALDH1A1KDM4EHPGDGLAGAA
Nitric Acid SCHEMBL3961222 0.79 KMT2A (0.49) ALDH1A1KDM4EHPGDGLAGAA
SCHEMBL31031113 0.77 NQO2 (0.49) ALDH1A1KDM4EGAAPOLBKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-106749185-A The synthesis of acridine esters chemical luminous substrate DMAENHS 湖南师范大学 2017-05-31 CN disclosed