SCHEMBL28147704

SCHEMBL28147704

C=C(C)C(=O)N(C)c1ccc(Br)cc1CN

nearest known ligand 0.33

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
POLB P06746 1/20 0.32
CYP2A6 P11509 1/20 0.32
ALDH1A1 P00352 1/20 0.32
STAT3 P40763 1/20 0.32
PDGFRA P16234 1/20 0.31
CDK5 Q00535 1/20 0.31
TYRO3 Q06418 1/20 0.31
SETDB1 Q15047 1/20 0.31
CCR5 P51681 1/20 0.31
NCEH1 Q6PIU2 1/20 0.31
SLC6A2 P23975 1/20 0.30
SLC6A4 P31645 1/20 0.30
SLC6A3 Q01959 1/20 0.30
CES1 P23141 1/20 0.30
PTGDR2 Q9Y5Y4 1/20 0.30
MEN1 O00255 1/20 0.30
KMT2A Q03164 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28356743 0.79 ALDH1A1 (0.36) POLBALDH1A1STAT3PDGFRACDK5
SCHEMBL28501470 0.78 ALDH1A1 (0.34) ALDH1A1STAT3PDGFRACDK5TYRO3
SCHEMBL31223908 0.74 XDH (0.33) ALDH1A1NCEH1MEN1KMT2A
SCHEMBL29213689 0.71 NOS3 (0.34) ALDH1A1NCEH1MEN1KMT2A
SCHEMBL27812573 0.70 PTGDR2 (0.39) CYP2A6ALDH1A1CCR5PTGDR2
SCHEMBL28353031 0.70 ALDH1A1 (0.40) POLBALDH1A1STAT3CES1MEN1
SCHEMBL27686826 0.68 ALDH1A1 (0.41) CYP2A6ALDH1A1CCR5MEN1KMT2A
SCHEMBL27593276 0.68 PTGDR2 (0.34) POLBCYP2A6ALDH1A1CCR5PTGDR2
SCHEMBL28995156 0.67 ALDH1A1 (0.36) ALDH1A1NCEH1
SCHEMBL28250213 0.66 KDM4E (0.37) POLBCYP2A6ALDH1A1MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-106749214-A Containing 1,3 benzoxazole difluoro methylene indole ketone compounds and preparation method thereof 上海大学 2017-05-31 CN disclosed